C07D 249/10
With hetero atoms or with carbon atoms having three bonds to hetero
Official title: with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
C07D249/10 (With hetero atoms or with carbon atoms having three bonds to hetero) appears on 1,798 US grants and 1,236 published applications in this corpus.
Search patents in C07D- Granted patents
- 1,798
- Published applications
- 1,236
- Assignees
- 661
- Inventors
- 4,430
- Latest grant
- 22 Sep 2026
Filings by year
| Year | Granted patents | Published applications |
|---|---|---|
| 1976 | 28 | 0 |
| 1977 | 25 | 0 |
| 1978 | 34 | 0 |
| 1979 | 25 | 0 |
| 1980 | 25 | 0 |
| 1981 | 38 | 0 |
| 1982 | 29 | 0 |
| 1983 | 27 | 0 |
| 1984 | 26 | 0 |
| 1985 | 20 | 0 |
| 1986 | 23 | 0 |
| 1987 | 24 | 0 |
| 1988 | 28 | 0 |
| 1989 | 30 | 0 |
| 1990 | 43 | 0 |
| 1991 | 45 | 0 |
| 1992 | 48 | 0 |
| 1993 | 52 | 0 |
| 1994 | 38 | 0 |
| 1995 | 42 | 0 |
| 1996 | 36 | 0 |
| 1997 | 35 | 0 |
| 1998 | 35 | 0 |
| 1999 | 40 | 0 |
| 2000 | 40 | 0 |
| 2001 | 53 | 10 |
| 2002 | 45 | 31 |
| 2003 | 46 | 55 |
| 2004 | 24 | 63 |
| 2005 | 31 | 52 |
| 2006 | 25 | 46 |
| 2007 | 24 | 38 |
| 2008 | 22 | 48 |
| 2009 | 25 | 45 |
| 2010 | 38 | 57 |
| 2011 | 37 | 59 |
| 2012 | 44 | 54 |
| 2013 | 48 | 62 |
| 2014 | 52 | 68 |
| 2015 | 56 | 71 |
| 2016 | 50 | 64 |
| 2017 | 50 | 61 |
| 2018 | 42 | 53 |
| 2019 | 41 | 50 |
| 2020 | 48 | 51 |
| 2021 | 42 | 50 |
| 2022 | 26 | 36 |
| 2023 | 30 | 35 |
| 2024 | 32 | 36 |
| 2025 | 18 | 23 |
| 2026 | 13 | 18 |
By publication year. Applications have been published since 2001. 2026 runs to 8 Oct.
Subgroups
Granted patents
Recent patents
- Headgroup lipid compounds and compositions for intracellular delivery of therapeutic agents22 Sep 2026US 12,740,943 B2ModernaTX, Inc.
- Agrochemical composition11 Aug 2026US 12,702,133 B2Upl Ltd
- Urea, amide, and substituted heteroaryl compounds for CBL-B inhibition16 Jun 2026US 12,653,809 B2Nurix Therapeutics, Inc.
- Aryl formamide compound containing chiral sulfur oxide or salt thereof, preparation method, herbicidal composition and use thereof2 Jun 2026US 12,643,871 B2Qingdao Kingagroot Chemical Compound Co., Ltd.
- [(5-phenyl-1-heteroaryl-1H-triazol-3-yl)oxy] acetic acid derivatives as safeners for the protection of useful plants and crop plants5 May 2026US 12,617,760 B2Bayer Aktiengesellschaft
- 3,5-diaminotriazole derivatives and uses thereof for treating ocular diseases24 Sep 2026US 2026/0284014 A1Centre National De La Recherche Scientifique
- At2 antagonists for non-addictive pain relief20 Aug 2026US 2026/0242357 A1Board of Regents, The University of Texas System
- Novel compounds6 Aug 2026US 2026/0226031 A1NRG Therapeutics Ltd
- Resist composition, resist pattern formation method, compound, and acid generator6 Aug 2026US 2026/0227692 A1Tokyo Ohka Kogyo.Co., Ltd.
- Compounds, compositions and uses thereof in the treatment and prevention of diseases and conditions associate with or aggravated by impaired mitophagy or oxidative stress30 Jul 2026US 2026/0217659 A1Yissum Research Development Company of the Hebrew University of Jerusalem
Most cited
By later US patents
- Nitrogen containing heteroaromatics as factor Xa inhibitors211US 6,020,357 ADuPont Pharmaceuticals Company · 2000
- Heterocyclic containing biphenyl aP2 inhibitors and method135US 6,548,529 B1Bristol-Myers Squibb Company · 2003
- Mutilin derivatives and their use as antibacterials115US 7,534,814 B2Nabriva Therapeutics AG · 2009
- Sulphonylaminocarbonyltriazolinones105US 5,625,074 ABayer Aktiengesellschaft · 1997
- Substituted 5-alkoxy-1,2,4-triazol-3-(THI) ones104US 5,652,372 ABayer Aktiengesellschaft · 1997