C07D 499/00
Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a
Official title: Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula: [IMAGE cpc-sch-C07D-0992.gif] , e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
C07D499/00 (Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a) appears on 1,115 US grants and 159 published applications in this corpus.
Search patents in C07D- Granted patents
- 1,115
- Published applications
- 159
- Assignees
- 280
- Inventors
- 1,419
- Latest grant
- 11 Aug 2026
Filings by year
| Year | Granted patents | Published applications |
|---|---|---|
| 1976 | 130 | 0 |
| 1977 | 84 | 0 |
| 1978 | 73 | 0 |
| 1979 | 44 | 0 |
| 1980 | 61 | 0 |
| 1981 | 60 | 0 |
| 1982 | 63 | 0 |
| 1983 | 51 | 0 |
| 1984 | 58 | 0 |
| 1985 | 54 | 0 |
| 1986 | 40 | 0 |
| 1987 | 34 | 0 |
| 1988 | 34 | 0 |
| 1989 | 42 | 0 |
| 1990 | 32 | 0 |
| 1991 | 20 | 0 |
| 1992 | 14 | 0 |
| 1993 | 13 | 0 |
| 1994 | 14 | 0 |
| 1995 | 8 | 0 |
| 1996 | 11 | 0 |
| 1997 | 25 | 0 |
| 1998 | 14 | 0 |
| 1999 | 10 | 0 |
| 2000 | 11 | 0 |
| 2001 | 6 | 1 |
| 2002 | 9 | 8 |
| 2003 | 3 | 7 |
| 2004 | 3 | 11 |
| 2005 | 3 | 9 |
| 2006 | 5 | 12 |
| 2007 | 3 | 5 |
| 2008 | 5 | 5 |
| 2009 | 3 | 12 |
| 2010 | 9 | 8 |
| 2011 | 1 | 3 |
| 2012 | 7 | 3 |
| 2013 | 4 | 7 |
| 2014 | 5 | 6 |
| 2015 | 3 | 4 |
| 2016 | 2 | 7 |
| 2017 | 4 | 5 |
| 2018 | 4 | 5 |
| 2019 | 4 | 7 |
| 2020 | 6 | 6 |
| 2021 | 6 | 9 |
| 2022 | 3 | 5 |
| 2023 | 5 | 3 |
| 2024 | 0 | 5 |
| 2025 | 8 | 5 |
| 2026 | 4 | 1 |
By publication year. Applications have been published since 2001. 2026 runs to 8 Oct.
Subgroups
Granted patents
- C07D 499/88Compounds with a double bond between positions 2 and 3 and a221
- C07D 499/21Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a70
- C07D 499/04Preparation22
- C07D 499/86Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a14
- C07D 499/897Compounds with substituents other than a carbon atom having three bonds to12
- C07D 499/87Compounds being unsubstituted in position 3 or with substituents other than only3
- C07D 499/90Further condensed with carbocyclic rings or ring systems1
Recent patents
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- Penem antibacterials against mycobacterial pathogens and d,d- and l,d transpeptidases11 Sep 2025US 2025/0282796 A1The Johns Hopkins University
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Most cited
By later US patents
- Pharmaceutical formulations for parenteral use208US 5,024,998 AUniversity of Florida · 1991
- 1,3-propane diol esters and ethers and methods for their use in drug delivery162US 6,555,700 B1Scotia Holdings PLC · 2003
- Fatty acid esters as bioactive compounds147US 6,245,811 B1Scotia Holdings PLC · 2001
- .beta.-Lactam antibacterial agents, their use in pharmaceutical compositions, and intermediates136US 4,282,236 ABeecham Group Limited · 1981
- Prodrug derivatives of carboxylic acid drugs122US 5,073,641 A1991