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US 9,040,457 B2Granted
Phenylamidines having a high fungicidal activity and use thereof
AssigneeIsagro S.p.A.
InventorsMarilena Gusmeroli, Lucio Filippini, Franco Pellacini, Paolo Bravini, Alexia Elmini, Matteo Santino Vazzola, Christian Badaracco
Life of this patent
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Abstract
New phenylamidines are described, having general formula (I): and their use for the control of phytopathogenic fungi.
Claims15
Phenylamidines having general formula (I):
- wherein
- R represents a phenyl, pyridyl, pyrimidyl, pyrazyl or pyridazyl group, wherein said phenyl, pyridyl, pyrimidyl, pyrazyl or pyridazyl group is substituted by at least a substituent selected from C1-C6 polyfluoroalkoxy containing at least one hydrogen atom, C1-C6 polyfluoroalkylthio containing at least one hydrogen atom, C3-C6 cycloalkyl, C3-C6 halocycloalkyl, C3-C6 cycloalkoxy, C3-C6 halocycloalkoxy, C4-C8 cycloalkylalkoxy, or C4-C8 halocycloalkylalkoxy;
- said phenyl, pyridyl, pyrimidyl, pyrazyl or pyridazyl being optionally substituted by one or two further substituents, equal to or different from each other, selected from halogen atom, C1-C6 alkyl, or C1-C6 haloalkyl;
- R1 represents C2-C6 alkyl;
- R2 represents C1-C6 alkyl;
- or R1 and R2, together with the N atom to which they are bound, form a heterocyclic ring containing from 4 to 7 atoms, optionally substituted by halogen atoms;
- R3 and R4, equal to or different from each other, represent a hydrogen atom, a halogen atom, a C1-C6 alkyl, a C1-C6 alkoxy, a C1-C6 haloalkoxy, a CF3 group, a CF2H group, a CFH2 group, or a cyano group.
4 more elements
A method for the control of phytopathogenic fungi of agricultural crops comprising applying an effective amount of a phenylamidine selected from general formula (I):
- wherein:
- R represents a phenyl, pyridyl, pyrimidyl, pyrazyl or pyridazyl group, wherein said phenyl, pyridyl, pyrimidyl, pyrazyl or pyridazyl group is substituted by at least a substituent selected from C1-C6 polyfluoroalkoxy containing at least one hydrogen atom, C1-C6 polyfluoroalkylthio containing at least one hydrogen atom, C3-C6 cycloalkyl, C3-C6 halocycloalkyl, C3-C6 cycloalkoxy, C3-C6 halocycloalkoxy, C4-C8 cycloalkylalkoxy, or C4-C8 halocycloalkylalkoxy;
- said groups phenyl, pyridyl, pyrimidyl, pyrazyl or pyridazyl being optionally substituted by one or two further substituents, equal to or different from each other, selected from halogen atom, C1-C6 alkyl, or C1-C6 haloalkyl;
- R1 represents C2-C6 alkyl;
- R2 represents C1-C6 alkyl;
- or R1 and R2, together with the N atom to which they are bound, form a heterocyclic ring containing from 4 to 7 atoms, optionally substituted by halogen atoms;
- R3 and R4, equal to or different from each other, represent a hydrogen atom, a halogen atom, C1-C6 alkyl, C1-C6 alkoxy, C1-C6 haloalkoxy, a CF3 group, a CF2H group, a CFH2 group, or a cyano group to phytopathogenic fungi of agricultural crops.
4 more elements
Dependencies are inferred from the claim text.