Back to results
US 8,785,630 B2Granted
Insecticidal triazines and pyrimidines
AssigneeVestaron Corporation
InventorsRobert M. Kennedy, Bruce A. Steinbaugh
Life of this patent
Estimating the term…
Abstract
The present invention describes novel triazines, their related pyrimidines and their use in controlling insects. This invention also includes new synthetic procedures, intermediates for preparing the compounds, pesticide compositions containing the compounds, and methods of controlling insects using the compounds.
Claims24
A method of using a compound of Formula (I),
- wherein:
- Y is CR1;
- R1 is —H, Halo or —C1-C4 alkyl;
- Z is -aryl, —C1-C8 alkylaryl, —C3-C8 cycloalkyl, —C1-C6 alkylC6cycloalkyl, heterocyclic, —C1-C8 alkylheterocyclic,
- X, is —H, —C1-C8 alkyl, -aryl, —C1-C8 alkylaryl, —C3-C8 cycloalkyl, —C1-C8 alkylC3-C8 cycloalkyl, heterocyclic, —C1-C8 alkylheterocyclic, —NRiRj or —C1-C8 alkylNRiRj;
- R2 and R3 are independently —H or —C1-C8 alkyl, -aryl, —C1-C8 alkylaryl, —C3-C8 cycloalkyl, —C1-C8 alkylC3-C8 cycloalkyl, heterocyclic, —C1-C8 alkylheterocyclic, and —C1-C8 alkylNRiRj, but R2 and R3 are not both H;
- Ri and Rj are independently —H, or —C1-C8 alkyl;
- wherein heterocyclic is a 5-10 member cyclic or bicyclic aromatic or saturated —C1-C8 cycloaliphatic ring moiety containing 1, 2, or 3 heteroatoms selected from N, O, or S;
- wherein aryl, —C3-C8 cycloalkyl and heterocyclic are optionally independently substituted with one to five substituents independently selected from -halo, —CN, —OH, —OCH2CH═CHCl, —C1-C6 alkyl, —O—C1-C6 alkyl, or —S—C1-C6 alkyl;
- and at each occurrence alkyl, is optionally substituted with 1-5 halo, —CN, or —OH in order to control and inhibit:
- insects, mites and nematodes, comprising applying an insect-inhibiting amount of a compound of Formula I to the locus, area to be protected or directly on the insects, mites and nematodes.
8 more elements
An insecticidal composition, with an optional phytologically-acceptable carrier comprising the compounds of Formula I, useful for the control of insects, mites and nematodes, where Formula I is:
- wherein:
- Y is N;
- R1 is —H, Halo or —C1-C4 alkyl;
- Z is -aryl, —C1-C8 alkylaryl, —C3-C8 cycloalkyl, —C1-C6 alkylC6cycloalkyl, heterocyclic, —C1-C8 alkylheterocyclic,
- X, is —H, —C1-C8 alkyl, -aryl, —C1-C8 alkylaryl, —C3-C8 cycloalkyl, —C1-C8 alkylC3-C8 cycloalkyl, heterocyclic, —C1-C8 alkylheterocyclic, —NRiRj or —C1-C8 alkylNRiRj;
- R2 and R3 are independently —H or —C1-C8 alkyl, -aryl, —C1-C8 alkylaryl, —C3-C8 cycloalkyl, —C1-C8 alkylC3-C8 cycloalkyl, heterocyclic, —C1-C8 alkylheterocyclic, and —C1-C8 alkylNRiRj, but R2 and R3 are not both H;
- Ri and Rj are independently —H, or —C1-C8 alkyl;
- wherein heterocyclic is a 5-10 member cyclic or bicyclic aromatic or saturated —C1-C8 cycloaliphatic ring moiety containing 1, 2, or 3 heteroatoms selected from N, O, or S;
- wherein aryl, —C3-C8 cycloalkyl and heterocyclic are optionally independently substituted with one to five substituents independently selected from -halo, —CN, —OH, —OCH2CH═CHCl, —C1-C6 alkyl, —O—C1-C6 alkyl, or —S—C1-C6 alkyl;
- and
- at each occurrence, alkyl is optionally substituted with 1-5 halo, —CN, or —OH.
8 more elements
Dependencies are inferred from the claim text.