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US 7,608,737 B2Granted
Naphthyl(ethyl)acetamides
AssigneeConcert Pharmaceuticasl Inc.
InventorsJulie F. Liu, Roger Tung
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Abstract
This disclosure relates to novel melatonin analogues or naphthyl(ethyl)acetamides, their derivatives, pharmaceutically acceptable salts, solvates, and hydrates thereof. This disclosure also provides compositions comprising a compound of this disclosure and the use of such compositions in methods of treating diseases and conditions that are beneficially treated by administering a dual melatoninergic agonist and serotoninergic antagonist.
Claims18
A compound of the Formula A:
- or a pharmaceutically acceptable salt, solvate or hydrate thereof, wherein:
- R1 is CD3;
- R2 is selected from OH, H, D and F;
- each of R3a, R3b, R4a, and R4b is independently selected from H and D;
- and
- R5is CD3.
3 more elements
Dependencies are inferred from the claim text.