US 7,408,008 B2Granted

Method of producing highly functionalized 1,3-diamino-propan-2-ols from solid support

AssigneeJanssen Pharmaceutica NV

InventorsSteve J. Coats, Dennis J. Hlasta, Mark J. Schulz

Life of this patent

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Abstract

The invention is directed to compounds and methods of synthesizing hydroxyethlamino amides and their use in treatment of aspartyl protease mediated diseases and conditions.

Claims3

Dependent claims

A compound of formula (Ia):

wherein (support) is selected from the group consisting of amine based polystyrene resins.

Dependencies are inferred from the claim text.

Facts

Application: 11/006,145Filed 7 Dec 2004 · us provisional application
Priority: 9 Dec 2003
Published: US 2005/0124001 A19 Jun 2005
Granted: 5 Aug 2008
Term ends: Not estimatedThe source records don’t support an estimate.

Classification29 codes

C07C 315/04
Preparation of sulfones; Preparation of sulfoxides: by reactions not involving the formation of sulfone or sulfoxide groups
C07C 233/37
With the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom: having the carbon atom of…
C07C 233/40
With the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom: having the carbon atom of…
C07C 233/62
Having carbon atoms of carboxamide groups bound to carbon atoms of rings other than six-membered aromatic rings: having the nitrogen atom of at…

Family

Application60/527,963Us provisional application · filed 9 Dec 2003
US 2005/0124001 A1Pre-grant publication · published 9 Jun 2005
US 7,408,008 B2This patent

From the US filing history. Foreign family members aren’t listed.

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