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US 5,708,183 AGranted
Process and intermediates for preparing triazolinones
AssigneeBayer Aktiengesellschaft
InventorHeinz-Jurgen Wroblowsky
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Abstract
The present invention relates to a novel process for preparing triazolinones of the general formula (I) ##STR1## in which R.sup.1 represents halogenoalkyl, and R.sup.2 represents hydrogen, hydroxyl or amino, or represents alkyl, alkenyl, alkinyl, alkoxy, alkylamino, dialkylamino, cycloalkyl, cycloalkylalkyl, phenyl or phenylalkyl which are in each case optionally substituted, and also to novel intermediates for preparing these triazolinones and to processes for preparing the intermediates themselves.
Claims2
A process for preparing a triazolinone of the formula (Ia):
- ##STR20## wherein R.sup.2 represents C.sub.1-6 -alkyl, C.sub.1-4 -alkoxy-C.sub.1-6 -alkyl, amino, C.sub.1-6 -alkylamino, or di-C.sub.1-6 -alkylamino;
- comprising cyclizing a hydrazinecarboxylic add ester of the formula (IIa):
- ##STR21## wherein R.sup.2 has the abovementioned meaning;
- and
- R represents C.sub.1-4 -alkyl, which is optionally substituted by halogen or C.sub.1-4 -alkoxy, or represents phenyl, which is optionally substituted by halogen or C.sub.1-4 -alkyl;
- or a tautomer of said hydrazinecarboxylic acid ester;
- in the presence of a base and a diluent at a temperature between 0.degree. C. and 150.degree. C.
4 more elements
Dependencies are inferred from the claim text.