Benzothiazine derivatives
AssigneeFujisawa Pharmaceutical Co., Ltd.
InventorsTsutomu Teraji, Teruo Oku, Youichi Shiokawa
Life of this patent
Estimating the term…
Loading patent…
AssigneeFujisawa Pharmaceutical Co., Ltd.
InventorsTsutomu Teraji, Teruo Oku, Youichi Shiokawa
Estimating the term…
This invention relates to novel benzothiazine derivatives having therapeutic effect on autoimmune diseases, to processes for preparation of such derivatives, and to pharmaceutical compositions containing such derivatives, the derivatives having the formula: ##STR1## wherein R.sup.1 is lower alkyl which may have one or more substituents selected from carboxy, aryl and carboxy(lower)cycloalkyl; aryl which may have one or more substituents selected from halogen, lower alkyl, halo(lower)alkyl and lower alkoxy; haloarylamino; or heterocyclic group; R.sup.2 is hydrogen, lower alkyl, lower alkylamino(lower)alkyl, aryl or ar(lower)alkyl; R.sup.3 is hydrogen, halogen, lower alkyl or lower alkoxy; and n is an integer 0 to 2.
A compound of the formula or its pharmaceutically acceptable salt:
Dependencies are inferred from the claim text.