1-Pyrrole- and 1-pyrrolidine-carboxylic acid derivatives and process for preparing the same
AssigneeLabaz
InventorsCharles Pigerol, Michel Schaefer, Souli Nanthavong
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AssigneeLabaz
InventorsCharles Pigerol, Michel Schaefer, Souli Nanthavong
Estimating the term…
1-Pyrrole- and 1-pyrrolidine-carboxylic acid derivatives corresponding to the general formula: ##STR1## in which R represents an alkyl radical having from 1 to 4 carbon atoms, preferably ethyl, and Am represents a group: ##STR2## wherein R.sub.1 represents a 3-oxo-alkyl radical ##STR3## or a 3-oxo-alkenyl radical ##STR4## and R.sub.2 represents hydrogen or R.sub.1 and R.sub.2, when they are identical, each represent hydrogen, ##STR5## R.sub.3 representing an alkyl radical having from 1 to 5 carbon atoms with the proviso that when R.sub.1 and R.sub.2 are simultaneously hydrogen, Am represents the group A. The novel derivatives are useful as intermediates for synthetizing azaprostaglandines.
2,5-Dihydro-1-pyrrole-carboxylic acid derivatives corresponding to the formula:
Ethyl 3-(1'-pyrrolidinyl)-2,5-dihydro-1-pyrrole-carboxylate.
Ethyl 4-(3'-oxo-butyl)-3-(1'-pyrrolidinyl)-2,5-dihydro-1-pyrrole-carboxylate.
Ethyl 4-(3'-oxo-butyl)-3-oxo-1-pyrrolidine-carboxylate.
Ethyl 4-(3'-oxo-octyl)-3-(1'-pyrrolidinyl)-2,5-dihydro-1-pyrrole-carboxylate.
Ethyl 4-(3'-oxo-octyl)-3-oxo-1-pyrrolidine-carboxylate.
Ethyl 4-(3'-oxo-1'-octenyl)-3-(1'-pyrrolidinyl)-2,5-dihydro-1-pyrrole-carboxylat e.
Ethyl 2,4-di-(3'-oxo-butyl)-3-(1'-pyrrolidinyl)-2,5-dihydro-1-pyrrole-carboxylat e.
Ethyl 2,4-di-(3'-oxo-butyl)-3-oxo-1-pyrrolidine-carboxylate.
Dependencies are inferred from the claim text.