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US 2024/0000075 A1Published application
Fungicidal aryl amidines
AssigneeCorteva Agriscience LLC
InventorsCRUZ AVILA-ADAME, VASUDEV R. BHONDE, SUSANA LOPEZ, BRIAN LOY, STACY T. MEYER, ALEX NOLAN, ADRIAN TLAHUEXT-ACA
Life of this patent
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Abstract
This disclosure relates to aryl amidines of Formula I and their use as fungicides.
Claims24
A compound of Formula I:
- wherein
- R1 is selected from the group consisting of C2-C8 alkyl, C1-C8 haloalkyl, C2-C8 alkenyl, C2-C8 substituted alkenyl, C2-C8 alkynyl, C2-C8 substituted alkynyl, C3-C8 cycloalkyl, C3-C8 substituted cycloalkyl, C3-C8 heterocycloalkyl, C3-C8 substituted heterocycloalkyl, C5-C7 heteroaryl, C5-C7 substituted heteroaryl, aryl, and substituted aryl;
- each R2 and R3 independently is selected from the group consisting of hydrogen, C1-C8 alkyl, C1-C8 haloalkyl, C2-C8 alkenyl, C2-C8 substituted alkenyl, C2-C8 alkynyl, C2-C8 substituted alkynyl;
- or R1 and R2 may be covalently bonded together to form a C4-C8 cycloalkyl group, C3-C8 substituted cycloalkyl group, C3-C8 heterocycloalkyl, or C3-C8 substituted heterocycloalkyl group;
- each R4, R5, and R6 independently is selected from the group consisting of hydrogen, halogen, cyano, nitro, C1-C8 alkyl, C1-C8 substituted alkyl, C2-C8 alkenyl, C2-C8 substituted alkenyl, C2-C8 alkynyl, C2-C8 substituted alkynyl, C1-C8 alkoxy, and C1-C8 substituted alkoxy;
- R7 is H;
- R8 is selected from the group consisting of hydrogen, C1-C8 alkyl, C1-C8 substituted alkyl, C2-C8 alkenyl, C2-C8 substituted alkenyl, C2-C8 alkynyl, C2-C8 substituted alkynyl, C1-C8alkoxy, and C1-C8 substituted alkoxy;
- or R8 and R9 may be covalently bonded together to form a C3-C8 heterocycloalkyl or C3-C8 substituted heterocycloalkyl group;
- each R9 and R10 independently is selected from the group consisting of C1-C8 alkyl, C1-C8 substituted alkyl, C2-C8 alkenyl, C2-C8 substituted alkenyl, C2-C8 alkynyl, C2-C8 substituted alkynyl, C3-C8 cycloalkyl, C3-C8 substituted cycloalkyl, aryl, substituted aryl, C1-C8 alkylaryl, and substituted C1-C8 alkylaryl;
- or R9 and R10 may be covalently bonded together to form a C3-C8 heterocycloalkyl or C3-C8 substituted heterocycloalkyl group;
- X is O;
- wherein any and all heterocyclic rings may contain up to three heteroatoms selected from the group consisting of O, N, and S;
- or a tautomer or salt thereof.
10 more elements
A compound wherein the compound is selected from one of the compounds in Table 1.
A fungicidal compound of Formula I.
- wherein
- R1 is selected from the group consisting of C2-C8 alkyl, C1-C8 haloalkyl, C2-C8 alkenyl, C2-C8 substituted alkenyl, C2-C8 alkynyl, C2-C8 substituted alkynyl, C3-C8 cycloalkyl, C3-C8 substituted cycloalkyl, C3-C8 heterocycloalkyl, C3-C8 substituted heterocycloalkyl, C5-C7 heteroaryl, C5-C7 substituted heteroaryl, aryl;
- and substituted aryl;
- each R2 and R3 independently is selected from the group consisting of hydrogen, C1-C8 alkyl, C1-C8 haloalkyl, C2-C8 alkenyl, C2-C8 substituted alkenyl, C2-C8 alkynyl, C2-C8 substituted alkynyl;
- or R1 and R2 may be covalently bonded together to form a C4-C8 cycloalkyl group, C3-C8 substituted cycloalkyl group, C3-C8 heterocycloalkyl, or C3-C8 substituted heterocycloalkyl group;
- each R4, R5, and R6 independently is selected from the group consisting of hydrogen, halogen, cyano, nitro, C1-C8 alkyl, C1-C8 substituted alkyl, C2-C8 alkenyl, C2-C8 substituted alkenyl, C2-C8 alkynyl, C2-C8 substituted alkynyl, C1-C8 alkoxy, and C1-C8 substituted alkoxy;
- R7 is H;
- R8 is selected from the group consisting of hydrogen, C1-C8 alkyl, C1-C8 substituted alkyl, C2-C8 alkenyl, C2-C8 substituted alkenyl, C2-C8 alkynyl, C2-C8 substituted alkynyl, C1-C8 alkoxy, C1-C8 substituted alkoxy, and thiol;
- or R8 and R9 may be covalently bonded together to form a C3-C8 heterocycloalkyl or C3-C8 substituted heterocycloalkyl group;
- each R9 and R10 independently is selected from the group consisting of C1-C8 alkyl, C1-C8 substituted alkyl, C2-C8 alkenyl, C2-C8 substituted alkenyl, C2-C8 alkynyl, C2-C8 substituted alkynyl, C3-C8 cycloalkyl, C3-C8 substituted cycloalkyl, aryl, substituted aryl, C1-C8 alkylaryl, and substituted C1-C8 alkylaryl;
- or R9 and R10 may be covalently bonded together to form a C3-C8 heterocycloalkyl or C3-C8 substituted heterocycloalkyl group;
- X is O;
- wherein any and all heterocyclic rings may contain up to three heteroatoms selected from the group consisting of O, N, and S;
- or a tautomer or salt thereof, for controlling a fungal pathogen.
11 more elements
Dependencies are inferred from the claim text.