US 2022/0264880 A1Published application

Novel heteroaryl-triazole compounds as pesticides

AssigneeBayer Aktiengesellschaft

InventorsAlexander ARLT, Hans-Georg SCHWARZ, Yolanda CANCHO GRANDE, Martin FUESSLEIN, Peter JESCHKE, Ulrich EBBINGHAUS-KINTSCHER, Marc LINKA, Peter LOESEL, Arunas Jonas DAMIJONAITIS, Andreas TURBERG, Iring HEISLER, Oleksandr MANDZHULO

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Abstract

The present invention relates to novel heteroaryl-triazole and heteroaryl-tetrazole compounds of the general formula (I), in which the structural elements R1, R2, R3, R4 and R5 have the meaning given in the description, to formulations and compositions comprising such compounds and for their use in the control of animal pests including arthropods and insects in plant protection and to their use for control of ectoparasites on animals.

Claims17

Dependent claims

A compound of formula (I)

in which
R1 is hydrogen;
R2 is phenyl wherein the phenyl is substituted with a total of one to two substituents, provided the substituent(s) are not on either carbon adjacent to the carbon bonded to the C═O group and one substituent is selected from group A consisting of
methylsulfonyl, ethylsulfonyl, isopropylsulfonyl, cyclopropylsulfonyl, difluoromethylsulfonyl, trifluoroethylsulfonyl, trifluoromethylsulfonyl, and —SF5 and cyclopropyl wherein the cyclopropyl is optionally substituted with one to two substituent(s) selected from the group of halogen, —CN, methyl, difluoromethyl and trifluoromethyl;
and the other substituent is independently selected from group B consisting of
fluorine, chlorine, bromine, iodine, —CN, difluoromethyl, trifluoromethyl, difluoromethoxy, trifluoromethoxy and cyclopropyl wherein the cyclopropyl is optionally substituted with one to two substituent(s) selected from the group of halogen, —CN, methyl, difluoromethyl and trifluoromethyl;
or
R2 is thiophene optionally substituted by one substituent selected from the group consisting of
fluorine, chlorine, bromine, and trifluoromethyl;
or
R2 is pyrazol optionally substituted by one to two substituents selected from the group consisting of
fluorine, chlorine, bromine, methyl, and trifluoromethyl;
R3 is C1-C3alkyl;
R4 is pyridine, pyrimidine or pyrazine wherein the pyridine, pyrimidine or pyrazine is optionally substituted with one substituent selected from the group consisting of
chlorine, and —CN;
R5 is ethyl, n-propyl, iso-propyl, difluoromethyl, cyclopropyl, methoxy, ethoxy, iso-propoxy or halogen.

13 more elements

Dependencies are inferred from the claim text.

Facts

Application: 17/628,519Filed 17 Jul 2020
Priority: EP 19187891.723 Jul 2019
Published: 25 Aug 2022
Term ends: Not estimatedThe source records don’t support an estimate.

Classification18 codes

A01N 43/653
Triazoles; Hydrogenated triazoles: 1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
A61K 45/06
Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00: mixtures of active ingredients without…
A01N 25/30
Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by…
A01N 43/54
Having rings with two nitrogen atoms as the only ring hetero atoms: 1,3-Diazines; Hydrogenated 1,3-diazines

Family

US 12,610,949 B2Related patent
US 2022/0264880 A1This patent

From the US filing history. Foreign family members aren’t listed.

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