Back to results
US 2010/0168217 A1Published application
Sulfamatobenzothiophene derivatives
AssigneeMerck Patent GmbH
InventorsWolfgang Staehle, David Bruge, Gerald Scholz, Benoit Rondot, Jean Lafay
Life of this patent
Estimating the term…
Abstract
The invention relates to novel compound of the general formula (I), in which R has the meanings indicated in claim 1, to the preparation thereof and to the use thereof as medicaments. The compounds (I) are inhibitors of steroid sulfatase and are used for the treatment of cancer.
Claims11
Compounds of the formula (I)
- in which
- R is a cycloalkyl ring having 3 to 12 C atoms or tert-butyl,
- R1 denotes H or alkyl having 1-6 C atoms,
- m denotes 0, 1, 2, 3 or 4
- n denotes 1 or 2,
- and pharmaceutically usable derivatives, salts, solvates and
- tautomers thereof, including mixtures thereof in all ratios.
4 more elements
Dependencies are inferred from the claim text.