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US 11,026,427 B2Granted
Microbiocidal oxadiazole derivatives
AssigneeSyngenta Participations AG
InventorsThomas James Hoffman, Daniel Stierli, Martin Pouliot
Life of this patent
Estimating the term…
Abstract
Compounds of the Formula (I), wherein the substituents are as defined in claim 1, useful as pesticides, especially as fungicides.
Claims13
A compound of formula (I):
- wherein
- A1 represents N or CR1, wherein R1 is hydrogen, halogen, methyl, ethyl, difluoromethyl, trifluoromethyl, methoxy, ethoxy or difluoromethoxy;
- A2 represents N or CR2, wherein R2 is hydrogen, halogen, methyl, ethyl, difluoromethyl, trifluoromethyl, methoxy, ethoxy or difluoromethoxy;
- A3 represents N or CR3, wherein R3 is hydrogen or fluoro;
- A4 represents N or CR4, wherein R4 is hydrogen or fluoro;
- and
- wherein no more than two of A1 to A4 are N;
- L1 represents —C(O)—;
- R5 represents cyano, cyanoC1-6alkyl, C1-3alkoxyC1-4alkyl, C1-2fluoroalkoxyC1-4alkyl, C3-6alkenyl, C3-6alkynyl, C3-8cycloalkyl or C3-8cycloalkylC1-2alkyl wherein the cycloalkyl moiety is optionally partially unsaturated, phenyl, phenylC1-2alkyl, heteroaryl bonded to L1 through a carbon atom or heteroarylC1-2alkyl, wherein the heteroaryl moiety is a 5- or 6-membered monocyclic aromatic ring which comprises 1, 2, 3 or 4 heteroatoms individually selected from N, O and S, heterocyclyl bonded to L1 through a carbon atom or heterocyclylC1-2alkyl, wherein the heterocyclyl moiety is a 4- to 6-membered non-aromatic ring which comprises 1, 2 or 3 heteroatoms individually selected from N, O and S, and wherein C3-8cycloalkyl, phenyl, heteroaryl and heterocyclyl are optionally substituted by 1, 2 or 3 substituents, which may be the same or different, selected from R7, and wherein when R5 represents C3-8cycloalkyl, C3-8cycloalkylC1-2alkyl, heterocyclyl or heterocyclylC1-2alkyl, the C3-8cycloalkyl or heterocyclyl moiety is optionally substituted by 1 or 2 oxo groups;
- R7 represents cyano, halogen, hydroxy, C1-4alkyl, C1-2haloalkyl, C1-4alkoxy, C1-2haloalkoxy, C1-4alkylcarbonyl, C1-4alkoxycarbonyl, aminocarbonyl, C1-4alkylaminocarbonyl or diC1-4alkylaminocarbonyl;
- or
- a salt or an N-oxide thereof.
9 more elements
A compound of formula (I):
- wherein
- A1 represents N or CR1, wherein R1 is hydrogen, halogen, methyl, ethyl, difluoromethyl, trifluoromethyl, methoxy, ethoxy or difluoromethoxy;
- A2 represents N or CR2, wherein R2 is hydrogen, halogen, methyl, ethyl, difluoromethyl, trifluoromethyl, methoxy, ethoxy or difluoromethoxy;
- A3 represents Nor CR3, wherein R3 is hydrogen or fluoro;
- A4 represents N or CR4, wherein R4 is hydrogen or fluoro;
- and
- wherein no more than two of A1 to A4 are N;
- L1 represents —C(OH)(R6)—;
- R5 represents cyano, C1-6haloalkyl, cyanoC1-6alkyl, C1-3alkoxyC1-4alkyl, C1-2fluoroalkoxyC1-4alkyl, C3-6alkenyl, C3-6alkynyl, C3-8cycloalkyl or C3-8cycloalkylC1-2alkyl wherein the cycloalkyl moiety is optionally partially unsaturated, phenyl, phenylC1-2alkyl, heteroaryl bonded to L1 through a carbon atom or heteroarylC1-2alkyl, wherein the heteroaryl moiety is a 5- or 6-membered monocyclic aromatic ring which comprises 1, 2, 3 or 4 heteroatoms individually selected from N, O and S, heterocyclyl bonded to L1 through a carbon atom or heterocyclylC1-2alkyl, wherein the heterocyclyl moiety is a 4- to 6-membered non-aromatic ring which comprises 1, 2 or 3 heteroatoms individually selected from N, O and S, and wherein C3-8cycloalkyl, phenyl, heteroaryl and heterocyclyl are optionally substituted by 1, 2 or 3 substituents, which may be the same or different, selected from R7, and wherein when R5 represents C3-8cycloalkyl, C3-8cycloalkylC1-2alkyl, heterocyclyl or heterocyclylC1-2alkyl, the C3-8cycloalkyl or heterocyclyl moiety is optionally substituted by 1 or 2 oxo groups;
- R6 represents hydrogen, C1-6alkyl, C3-6alkenyl, C3-6alkynyl or C1-2haloalkyl;
- R7 represents cyano, halogen, hydroxy, C1-4alkyl, C1-2haloalkyl, C1-4alkoxy, C1-2haloalkoxy, C1-4alkylcarbonyl, C1-4alkoxycarbonyl, aminocarbonyl, C1-4alkylaminocarbonyl or diC1-4alkylaminocarbonyl;
- or
- a salt or an N-oxide thereof.
10 more elements
Dependencies are inferred from the claim text.