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US 10,501,441 B2Granted
Substituted imidazolylcarboxamides as pesticides
AssigneeBayer CropScience AG
InventorsMarkus Heil, Reiner Fischer, Johannes-Rudolf Jansen, David Wilcke, Matthieu Willot, Susanne Kübbeler, Kerstin Ilg, Sascha Eilmus, Peter Lösel, Wolfram Andersch, Ulrich Görgens
Life of this patent
Estimating the term…
Abstract
The present invention relates to compounds of the general formula (I) in which Q, V, T, W, Y, L1, L2 and A have the meanings given in the description—and to their use for controlling animal pests.
Claims14
Compound of formula (I)
- in which
- Q represents oxygen or sulphur,
- V represents a radical from the group consisting of hydrogen, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy and cyano,
- W represents a radical from the group consisting of hydrogen, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy and cyano,
- Y represents a radical from the group consisting of hydrogen, cyano, optionally substituted alkyl, alkenyl or alkynyl, optionally substituted cycloalkyl which is optionally interrupted by heteroatoms, optionally substituted cycloalkylalkyl which is optionally interrupted by heteroatoms, arylalkyl or hetarylalkyl,
- A represents a radical from the group consisting of hydrogen, optionally substituted alkyl, alkenyl or alkynyl and optionally substituted cycloalkyl or cycloalkylalkyl which are optionally interrupted by heteroatoms,
- T represents oxygen or an electron pair,
- L1 represents a radical from the group consisting of hydrogen, optionally substituted alkyl, alkenyl, alkynyl, or cycloalkyl and represents the radicals C(O)R2, C(O)N(R3)(R4), C(O)OR5 and SO2R6,
- L2 represents a radical from the group consisting of hydrogen, N(R3a)(R4a), optionally substituted alkyl, alkenyl, alkynyl or alkoxy, optionally substituted cycloalkyl or cycloalkylalkyl which is optionally interrupted by heteroatoms, and optionally substituted aryl, arylalkyl, hetaryl or hetarylalkyl,
- or
- L1 and L2 represent, together with the nitrogen atom to which they are attached, an optionally substituted saturated, partially saturated or aromatic heterocycle having 3 to 7 ring atoms which can optionally be interrupted by further heteroatoms and/or by one or two C═O groups,
- R2 represents a radical from the group consisting of hydrogen, optionally substituted alkyl, alkenyl or alkynyl, optionally substituted cycloalkyl, optionally substituted aryl or hetaryl and optionally substituted arylalkyl or hetarylalkyl,
- R3 and R4 each independently of one another represent a radical from the group consisting of hydrogen, optionally substituted alkyl, alkenyl or alkynyl, optionally substituted saturated or unsaturated cycloalkyl, cycloalkylalkyl, aryl, hetaryl, arylalkyl or hetarylalkyl,
- or
- R3 and R4 together form an optionally substituted three- to seven-membered aliphatic ring which optionally contains a nitrogen, sulphur or oxygen atom,
- R3a represents a radical from the group consisting of hydrogen, optionally substituted alkyl, optionally substituted cycloalkyl, aryl, hetaryl, arylalkyl or hetarylalkyl,
- R4a represents a radical from the group consisting of hydrogen, optionally substituted alkyl, optionally substituted C3-C6-cycloalkyl and represents the radicals C(O)R2, C(O)OR5 and SO2R6,
- R5 represents optionally substituted alkyl, alkenyl or alkynyl, optionally substituted cycloalkyl or cycloalkylalkyl,
- R6 represents a radical from the group consisting of optionally substituted alkyl, alkenyl or alkynyl, optionally substituted cycloalkyl cycloalkylalkyl, aryl, arylalkyl, hetaryl or hetarylalkyl
- And/or a salt thereof.
17 more elements
Intermediate of formula (VI)
- Wherein
- Q represents oxygen or sulphur,
- V represents a radical from the group consisting of hydrogen, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy and cyano,
- W represents a radical from the group consisting of hydrogen, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy and cyano,
- Y represents a radical from the group consisting of hydrogen, cyano, optionally substituted alkyl, alkenyl or alkynyl, optionally substituted cycloalkyl which is optionally interrupted by heteroatoms, optionally substituted cycloalkylalkyl which is optionally interrupted by heteroatoms, arylalkyl or hetarylalkyl,
- A represents a radical from the group consisting of hydrogen, optionally substituted alkyl, alkenyl or alkynyl and optionally substituted cycloalkyl or cycloalkylalkyl which are optionally interrupted by heteroatoms,
- T represents oxygen or an electron pair,
- L1 represents a radical from the group consisting of hydrogen, optionally substituted alkyl, alkenyl, alkynyl, or cycloalkyl and represents the radicals C(O)R2, C(O)N(R3)(R4), C(O)OR5 and SO2R6,
- L2 represents a radical from the group consisting of hydrogen, N(R3a)(R4a), optionally substituted alkyl, alkenyl, alkynyl or alkoxy, optionally substituted cycloalkyl or cycloalkylalkyl which is optionally interrupted by heteroatoms, and optionally substituted aryl, arylalkyl, hetaryl or hetarylalkyl,
- or
- L1 and L2 represent, together with the nitrogen atom to which they are attached, an optionally substituted saturated, partially saturated or aromatic heterocycle having 3 to 7 ring atoms which can optionally be interrupted by further heteroatoms and/or by one or two C═O groups,
- R2 represents a radical from the group consisting of hydrogen, optionally substituted alkyl, alkenyl or alkynyl, optionally substituted cycloalkyl, optionally substituted aryl or hetaryl and optionally substituted arylalkyl or hetarylalkyl,
- R3 and R4 each independently of one another represent a radical from the group consisting of hydrogen, optionally substituted alkyl, alkenyl or alkynyl, optionally substituted saturated or unsaturated cycloalkyl, cycloalkylalkyl, aryl, hetaryl, arylalkyl or hetarylalkyl,
- or
- R3 and R4 together form an optionally substituted three- to seven-membered aliphatic ring which optionally contains a nitrogen, sulphur or oxygen atom,
- R3a represents a radical from the group consisting of hydrogen, optionally substituted alkyl, optionally substituted cycloalkyl, aryl, hetaryl, arylalkyl or hetarylalkyl,
- R4a represents a radical from the group consisting of hydrogen, optionally substituted alkyl, optionally substituted C3-C6-cycloalkyl and represents the radicals C(O)R2, C(O)OR5 and SO2R6,
- R5 represents optionally substituted alkyl, alkenyl or alkynyl, optionally substituted cycloalkyl or cycloalkylalkyl,
- R6 represents a radical from the group consisting of optionally substituted alkyl, alkenyl or alkynyl, optionally substituted cycloalkyl cycloalkylalkyl, aryl, arylalkyl, hetaryl or hetarylalkyl
- and/or a salt thereof.
17 more elements
Dependencies are inferred from the claim text.