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US 9,067,930 B2Granted
2-oxo-piperidinyl derivatives
AssigneeUCB Pharma S.A.
InventorsAli Ates, Florian Montel, Anne Valade, Olivier Lorthioir
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Abstract
The present invention relates to 2-oxo-piperidinyl derivatives, processes for preparing them, pharmaceutical compositions containing them and their use as pharmaceuticals.
Claims11
A 2-Oxo-piperidinyl compound of the form according to formula I, or a geometrical isomer, enantiomer, diastereomer or mixture, or a pharmaceutically acceptable salt thereof,
- wherein
- X is either CH or N;
- Y is either —NR4— or —CH═CH—;
- with the proviso that X is N when Y is —NR4—;
- n is an integer selected from 1, 2 or 3;
- m is 1 or 2;
- R1 is a substituted or unsubstituted C1-6 alkyl, a substituted or unsubstituted aryl, a substituted or unsubstituted heterocycle, a substituted or unsubstituted C3-8 cycloalkyl;
- or R1 is a —O—R2 moiety;
- R2 is a substituted or unsubstituted C1-6 alkyl, a substituted or unsubstituted aryl or a substituted or unsubstituted heteroaryl;
- R3 is hydrogen, substituted or unsubstituted C1-4 alkyl or halogen;
- and
- R4 is hydrogen or C1-4 alkyl.
9 more elements
Dependencies are inferred from the claim text.