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US 8,895,534 B2Granted
Boron containing small molecules
AssigneeAnacor Pharmaceuticals, Inc.
InventorsStephen J. Baker, Vincent S. Hernandez, Rashmi Sharma, James A. Nieman, Tsutomu Akama, Yong-Kang Zhang, Jacob J. Plattner, Michael Richard Kevin Alley, Rajeshwar Singh, Fernando Rock
Life of this patent
Estimating the term…
Abstract
Novel monosubstituted and disubstutituted oxaboroles and pharmaceutical compositions containing such oxaboroles are provided, which are useful for treating bacterial infections, as well as combinations of these oxaboroles with at least one additional therapeutically effective agent.
Claims29
A compound having a structure according to the formula:
- wherein
- R* is H;
- R3 is —CH2NH2;
- Ra is H or —YR5
- wherein
- Y is O;
- R5 is:
- wherein
- a is an integer selected from 1, 2, 3, or 4;
- each R10 and each R11 is H;
- R12 is H;
- or a salt thereof.
9 more elements
A compound having a structure which is:
- or a salt thereof.
A compound which is
- or a salt thereof.
A compound which is
- or a salt thereof.
A compound which is
- or a salt thereof.
A compound which is
- or a salt thereof.
Dependencies are inferred from the claim text.