Inhibitors of histone deacetylase
AssigneeMethylGene Inc.
InventorsTammy Mallais, Oscar Moradei, Alain Ajamian, Pierre Tessier, David Smil, Sylvie Frechette, Silvana Leit, Patrick Beaulieu, Robert Deziel, John Mancuso
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Abstract
This invention relates to compounds and methods for the inhibition of HDAC enzymatic activity. More particularly, the invention provides for compounds of formula (I), (I) and N-oxides, hydrates, solvates, pharmaceutically acceptable salts, prodrugs and complexes thereof, and racemic and scalemic mixtures, diastereomers and enantiomers thereof, wherein L, M, n, R, W, X and Y are as defined in the specification.
Claims2
A compound or an N-oxide, hydrate, solvate, pharmaceutically acceptable salt, prodrug or complex thereof, in the form of a racemic or scalemic mixture, tautomer, diastereomer or enantiomer thereof, wherein the compound is selected from,
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Dependencies are inferred from the claim text.