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US 8,557,821 B2Granted
Microbiocidal heterocycles
AssigneeSyngenta Crop Protection AG
InventorsSarah Sulzer-Mosse, Clemens Lamberth, Mathias Stephan Respondek, Laura Quaranta
Life of this patent
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Abstract
The present invention relates to heterocyclic compounds of formula (I) which have microbiocidal activity, in particular fungicidal activity, as well as methods of using the compounds of formula (I) to control microbes.
Claims15
A compound of formula I:
- wherein
- A is x-C(═O)—, x-C(═S)—, x-C(R10R11)—C(═O)—, x-C(R12R13)—C(═S)—, x-O—C(═O)—, x-O—C(═S)—, x-N(R14)—C(═O)—, x-N(R15)—C(═S)—, x-C(R16R17)—SO2— or x-N═C(R26)—,in each case x indicates the bond that is connected to R1;
- T is CR18 or N;
- G is O or S;
- Y1 and Y2 are independently CR19 or N;
- Q is —C(═O)-z, —C(═S)-z, —C(═O)—O-z, —C(═S)—O-z, —C(═O)—N(R20)-z, —C(═S)—N(R21)-z or —SO2-z-, in each case z indicates the bond that is connected to R9;
- n is 1 or 2;
- p is 1 or 2, providing that when n is 2, p is 1;
- R1 is phenyl, pyridyl, imidazolyl, or pyrazolyl;
- wherein the phenyl, pyridyl, imidazolyl and pyrazolyl are each optionally substituted by 1 to 3 substituents independently selected from C1-C4 alkyl, C1-C4 haloalkyl, halogen, cyano, hydroxy and amino;
- R2, R3, R4, R5, R6, R7, R10, R11, R12, R13, R16, R17, R18, R19 and R26 each independently are hydrogen, halogen, cyano, C1-C4 alkyl or C1-C4haloalkyl;
- R8, R14, R15, R20 and R21 each independently are hydrogen, C1-C4 alkyl or C1-C4alkoxy;
- and
- R9 is phenyl, benzyl or group (a):
- wherein the phenyl, benzyl and group (a) are each optionally substituted with 1 to 3 substituents independently selected from C1-C4 alkyl, C1-C4 haloalkyl, C1-C4 alkoxy, C1-C4 haloalkoxy, halogen, cyano, hydroxyl, N(R27)2, SH, C1-C4 alkylthio, nitro, phenylsulfonyl and phenylsulfinyl, wherein the phenylsulfonyl and phenylsulfinyl are optionally substituted by 1 to 3 substituents independently selected from C1-C4 alkyl, C1-C4 haloalkyl, C1-C4 alkoxy, C1-C4 haloalkoxy, halogen and cyano;
- each R27 independently is hydrogen, C1-C4 alkyl, phenylsulfonyl or phenylsulfinyl, wherein the phenylsulfonyl and phenylsulfinyl are optionally substituted by 1 to 3 substituents independently selected from C1-C4 alkyl, C1-C4 haloalkyl, C1-C4 alkoxy, C1-C4 haloalkoxy, halogen and cyano;
- or a salt or a N-oxide thereof.
14 more elements
A compound of formula I.a:
- in which R1′ is C1-C8 alkyl
- or a compound of formula II:
- or a compound of formula VIII:
Dependencies are inferred from the claim text.