Antibacterial agents
AssigneeOptimer Pharmaceuticals, Inc.
InventorsJonathan Duffield, Chan-Kou Hwang, Yoshitaka Ichikawa, Youe-Kong Shue
Life of this patent
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Abstract
Described herein are novel macrolides, the preparation of novel macrolides, the use of novel macrolides for preventing, treating, or ameliorating various conditions, and the use of novel macrolides as antibacterial agents.
Claims25
A compound of the formula
- or a pharmaceutically acceptable salt or hydrate thereof, wherein:
- A is —CH2—;
- B is —(CH2)n—, where n is an integer in the range from 0 to 10;
- C is aryl or heteroaryl;
- and
- W is H or F.
A pharmaceutical composition comprising an anti-bacterially effective amount of a compound of the formula
- wherein:
- A is —CH2—;
- B is —(CH2)n—, where n is an integer in the range from 0 to 10;
- C is aryl or heteroaryl;
- and
- W is H or F.
A compound of the formula
- or a pharmaceutically acceptable salt or hydrate thereof.
A pharmaceutical composition comprising an anti-bacterially effective amount of a compound of the formula
A compound of the formula
- or a pharmaceutically acceptable salt thereof.
A pharmaceutical composition comprising a compound of the formula,
- or a pharmaceutically acceptable salt thereof, and a physiologically acceptable carrier or excipient.
Dependencies are inferred from the claim text.