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US 7,803,797 B2Granted
Substituted arylcyclopentenes as therapeutic agents
AssigneeAllergan, Inc.
InventorsDavid W. Old, Vinh X. Ngo
Life of this patent
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Abstract
Compounds comprising or a pharmaceutically acceptable salt or a prodrug thereof, are disclosed, wherein G, B, Y, and A are as described. Methods, compositions, and medicaments related thereto are also disclosed.
Claims11
A compound of the formula
- or a pharmaceutically acceptable salt thereof or a prodrug thereof;
- wherein Y is
- A is —(CH2)6—, cis —CH2CH═CH—(CH2)3—, or —CH2C≡C—(CH2)3—, wherein 1 or 2 carbon atoms may be replaced by S or O;
- or A is —(CH2)m—Ar—(CH2)o— wherein Ar is interarylene or heterointerarylene, the sum of m and o is 1, 2, 3, or 4, and wherein 1 —CH2— may be replaced by S or O, and 1 —CH2—CH2— may be replaced by —CH═CH— or —C═C—;
- G is H or OH;
- and
- B is aryl or heteroaryl.
4 more elements
Dependencies are inferred from the claim text.