US 7,683,070 B2 · N-(substituted arylmethyl)-4-(disubstituted methyl) piperidines and pyridines

N-(substituted arylmethyl)-4-(disubstituted methyl) piperidines and pyridines

AssigneeFMC Corporation

InventorsPing Ding, Robert N. Henrie, II, Daniel H. Cohen, John W. Lyga, David S. Rosen, George Theodoridis, Qun Zhang, Walter H. Yeager, Stephen F. Donovan, Stephen Shunxiang Zhang, Inna Shulman, Seong Jae Yu, Guozhi Wang, Y. Larry Zhang, Ariamala Gopalsamy, Dennis L. Warkentin, Paul E. Rensner, Ian R. Silverman, Thomas G. Cullen

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Abstract

It has now been found that certain novel N-(substituted aryl)-4-(disubstituted methyl)piperidine and pyridine derivatives have provided unexpected insecticidal activity. These compounds are represented by formula (I): wherein m, n, q, r, and s are independently selected from 0 or 1; and p is 0, 1, 2, or 3; A is C or CH; and B, D, E, R, R1, R2, R3, R4, R5, R6, R7 and R8 are fully described herein. In addition, compositions comprising an insecticidally effective amount of at least one compound of formula I, and optionally, an effective amount of at least one of a second compound, with at least one insecticidally compatible carrier are also disclosed; along with methods of controlling insects comprising applying said compositions to a locus where insects are present or are expected to be present.

Claims6

Dependent claims

A compound of formula I

wherein;
p, q, and rare 0;
s is 1;
A is C forming 1,2,5,6-tetrahydropyridine;
R2, R3, R4, R5, and R6 are independently selected from hydrogen, halogen, alkyl, and haloalkyl;
B is phenyl substituted with R9, R10, R11, R12, and R13,
where
R9, R10, R11, R12, and R13 are independently selected from hydrogen, halogen, alkyl, or haloalkyl;
R8 is phenyl substituted with R22, R23, R24, R25, and R26,
where
R22, R23, R25, and R26 are independently selected from hydrogen, alkyl, hydroxy, or alkoxy;
is an optionally substituted heteroaryloxy moiety;
E is (CR27R28)x—(CR29R30)y;
where
x is 1;
y is 0;
and,
where R27, R28, R29, and R30 are independently selected from hydrogen or alkyl;
and
agriculturally-acceptable salts thereof.

17 more elements

Dependencies are inferred from the claim text.

Facts

Application

11/874,015Filed 17 Oct 2007 · division

Priority

18 Dec 2002

Published

US 2008/0090828 A117 Apr 2008

Granted

23 Mar 2010

Term ends

Not estimatedThe source records don’t support an estimate.

Classification25 codes

C07D 405/14
Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having…:…
A01N 43/40
Having rings with one nitrogen atom as the only ring hetero atom: six-membered rings
A01N 43/54
Having rings with two nitrogen atoms as the only ring hetero atoms: 1,3-Diazines; Hydrogenated 1,3-diazines
A01N 43/713
Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds: having rings with four or more nitrogen…

Family

Application60/434,718Us provisional application · filed 18 Dec 2002

Application60/495,059Us provisional application · filed 14 Aug 2003

PCT/US2003/038878Parent of this division · filed 8 Dec 2003

US 2008/0090828 A1Pre-grant publication · published 17 Apr 2008

Application10/538,998Parent of this division

US 7,300,946 B2Parent of this division

US 2006/0135504 A1Published application

US 7,683,070 B2This patent

From the US filing history. Foreign family members aren’t listed.