Back to results
US 7,598,389 B2Granted
Silylated carboxamides
AssigneeBayer CropScience AG
InventorsRalf Dunkel, Hans-Ludwig Elbe, Benoit Hartmann, Alexander Klausener, Jörg Nico Greul, Ulrike Wachendorff-Neumann, Peter Dahmen, Karl-Heinz Kuck
Life of this patent
Estimating the term…
Abstract
Novel silylated carboxamides of the formula (I) in which R, L, R1, R3, R3, R4 and A are as defined in the description, a plurality of processes for preparing these compounds and their use for controlling unwanted microorganisms.
Claims15
Silylated carboxamides of the formula (I)
- in which
- R is hydrogen, fluorine, chlorine, methyl, isopropyl, methylthio or trifluoro-methyl,
- L is a direct bond or is in each case optionally substituted straight-chain or branched alkylene (alkanediyl), alkenylene (alkenediyl) or alkynylene (alkyndiyl),
- R1 and R2 independently of one another are hydrogen, C1-C8-alkyl, C1-C8-alkoxy, C1-C4-alkoxy-C1-C4-alkyl, C1-C4-alkylthio-C1-C4-alkyl or C1-C6-haloalkyl,
- R3 is hydrogen, C1-C8-alkyl, C1-C8-alkoxy, C1-C4-alkoxy-C1-C4-alkyl, C1-C4-alkylthio-C1-C4-alkyl, C2-C8-alkenyl, C2-C8-alkynyl, C1-C6-haloalkyl, C2-C6-halo-alkenyl, C2-C6-haloalkynyl, C3-C6-cycloalkyl, or is in each case optionally substituted phenyl or phenylalkyl,
- R4 is hydrogen, C1-C8-alkyl, C1-C6-alkylsulphinyl, C1-C6-alkylsulphonyl, C1-C4-alkoxy-C1-C4-alkyl, C3-C8-cycloalkyl;
- C1-C6-haloalkyl, C1-C4-haloalkylthio, C1-C4-haloalkylsulphinyl, C1-C4-haloalkylsulphonyl, halo -C1-C4-alkoxy-C1-C4-alkyl, C3-C8-halocycloalkyl having in each case 1 to 9 fluorine, chlorine and/or bromine atoms;
- formyl, formyl-C1-C3-alkyl, (C1-C3-alkyl)carbonyl-C1-C3-alkyl, (C1-C3-alkoxy)carbonyl-C1-C3-alkyl;
- halo-(C1-C3-alkyl)carbonyl-C1-C3-alkyl, halo-(C1-C3-alkoxy)carbonyl-C1-C3-alkyl having in each case 1 to 13 fluorine, chlorine and/or bromine atoms;
- (C1-C8-alkyl)carbonyl, (C1-C8-alkoxy)carbonyl, (C1-C4-alkoxy-C1-C4-alkyl)carbonyl, (C3-C8-cycloalkyl)carbonyl;
- (C1-C6-haloalkyl)carbonyl, (C1-C6-halo-alkoxy)carbonyl, (halo-C1-C4-alkoxy-C1-C4-alkyl)carbonyl, (C3-C8-halocyclo-alkyl)carbonyl having in each case 1 to 9 fluorine, chlorine and/or bromine atoms;
- or —C(═O)C(═O)R5, —CONR6R7 or —CH2NR8R9,
- R5 is hydrogen, C1-C8-alkyl, C1-C8-alkoxy, C1-C4-alkoxy-C1-C4-alkyl, C3-C8-cycloalkyl;
- C1-C6-haloalkyl, C1-C6-haloalkoxy, halo-C1-C4-alkoxy-C1-C4-alkyl, C3-C8-halocycloalkyl having in each case 1 to 9 fluorine, chlorine and/or bromine atoms,
- R6 and R7 independently of one another each are hydrogen, C1-C8-alkyl, C1-C4-alkoxy-C1-C4-alkyl, C3-C8-cycloalkyl;
- C1-C8-haloalkyl, halo-C1-C4-alkoxy-C1-C4-alkyl, C3-C8-halocycloalkyl having in each case 1 to 9 fluorine, chlorine and/or bromine atoms,
- R6 and R7 furthermore together with the nitrogen atom to which they are attached form a saturated heterocycle having 5 to 8 ring atoms which is optionally mono- or polysubstituted by identical or different substituents from the group consisting of halogen and C1-C4-alkyl, where the heterocycle may contain 1 or 2 further nonadjacent heteroatoms from the group consisting of oxygen, sulphur and NR10,
- R8 and R9 independently of one another, are hydrogen, C1-C8-alkyl, C3-C8-cycloalkyl;
- C1-C8-haloalkyl, C3-C8-halocycloalkyl having in each case 1 to 9 fluorine, chlorine and/or bromine atoms,
- R8 and R9 furthermore together with the nitrogen atom to which they are attached form a saturated heterocycle having 5 to 8 ring atoms which is optionally mono- or polysubstituted by identical or different substituents from the group consisting of halogen and C1-C4-alkyl, where the heterocycle may contain 1 or 2 further nonadjacent heteroatoms from the group consisting of oxygen, sulphur and NR10,
- R10 is hydrogen or C-1-C6-alkyl,
- A is the radical of the formula (A2)
- R12 is chlorine or iodine.
20 more elements
Dependencies are inferred from the claim text.