Analgesics, anaesthetics, antifoulants, aversants, irritants, incapacitants and compositions containing the same
AssigneeWhite Flower Associates LLP
InventorMel Blum
Life of this patent
Estimating the term…
Abstract
Compounds and compositions the same. Method of making the compounds. The compounds and/or compositions used as an analgesic, anaesthetic, antifoulant, aversant, irritant, sternutator, neurodegenerator, counter irritant (delayed), rubifaciant, stomachic, fungicide, insecticide, preservative, circulatory stimulant, cardio-protective agent, immune booster, decongestant, anti-inflammatory agent, incapacitant, biocide, mildewcide, pharmaceutical, repellent, flavorant, carminative, antismoking agent, and/or antithrombotic agent. One of the compounds being lidocaine nonivamide. The compositions comprising one or more of: the compounds, one or more of an antioxidant, a UV absorber, and one or more biocides such as, for example, OBPA.
Claims33
A compound selected from the group consisting of:
- lidocaine nonivamide, benzocaine nonivamide, butacaine nonivamide, dibucaine nonivamide, procaine nonivamide, tetracaine nonivamide, lidocaine capsaicinate, benzocaine capsaicinate, butacaine capsaicinate, dibucaine capsaicinate, procaine capsaicinate, and tetracaine capsaicinate.
A method for the production of novel compounds, comprising:
- providing hydrochlorides of one or more of the following compounds:
- lidocaine, benzocaine, butacaine, dibucaine, procaine, and tetracaine,
- converting said hydrochlorides of said one or more compounds to hydroxides of said one or more compounds;
- and
- reacting said hydroxides of said one or more compounds with capsaicin and/or nonivamide.
A method for the production of novel compounds, comprising:
- reacting benzocaine with nonivamide and/or capsaicin.
A composition comprising nonivamide and OBPA.
Dependencies are inferred from the claim text.