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US 7,396,943 B2Granted
Opioid receptor antagonists
AssigneeEli Lilly and Company
InventorsDana Rae Benesh, Maria Jesus Blanco-Pillado, Charles Howard Mitch, Kumiko Takeuchi
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Abstract
A compound of the formula I: (I) wherein the variables are as described herein, or a pharmaceutically acceptable salt, solvate, enantiomer, racemate, diastereomer or mixture thereof, formulations and methods of use thereof are disclosed.
Claims2
A compound selected from the group consisting of:
- 4-[5-(Phenethylamino-methyl)-thiophen-2-yloxy]-benzamide
- 4-{5-[(3-Methyl-butylamino)-methyl]-thiophen-2-yloxy}-benzamide
- 4-(5-{[2-(3-Fluoro-phenyl)-ethylamino]-methyl}-thiophen-2-yloxy)-benzamide
- 4-{5-[(2-Cyclopentyl-ethylamino)-methyl]-thiophen-2-yloxy}-benzamide
- 4-{5-[(2-Thiophen-2-yl-ethylamino)-methyl]-thiophen-2-yloxy}-benzamide
- 4-{5-[(3,3-Dimethyl-butylamino)-methyl]-thiophen-2-yloxy}-benzamide
- 3-Methoxy-4-[5-(phenethylamino-methyl)-thiophen-2-yloxy]-benzamide
- 3-Methoxy-4-{5-[(3-methyl-butylamino)-methyl]-thiophen-2-yloxy}-benzamide
- 4-[5-(2-Phenethylamino-ethyl)-thiophen-2-yloxy]-benzamide
- 5-{4-[(3-Ethylpentylamino)methyl]phenoxy}thiophene-2-carboxamide
- 2-{4-[(3-Methylbutylamino)methyl]phenoxy}thiazole-5-carboxamide
- 2-(4-{[2-(Tetrahydropyran-4-yl)ethylamino]methyl}phenoxy)thiazole-5-carboxamide
- or a pharmaceutically acceptable salt thereof.
10 more elements
Dependencies are inferred from the claim text.