Mercaptophenyl naphthyl methane compounds and synthesis thereof

A mercaptophenyl naphthyl methane compound having the structural formula 1:

• wherein R is CHOH, wherein R1 is H or C1-C6-alkyl, wherein R2 is H or C1-C6 alkyl and wherein R3 is selected from the group consisting of H, or C1-C6 alkyl, and wherein R3 is SR6 or SO2R6, wherein R6 is selected from the group consisting of H, C1-C6 alkyl, aminoalkyl, pyrrolidinoethyl, piperidinoethyl, dimenthylaminoethyl, and diethylaminoethyl.

A pharmaceutical composition comprising a mercaptophenyl naphthyl methane compound having structural formula 1

• wherein R is CHOH, wherein R1 is H or C1-C6-alkyl, wherein R2 is H or C1-C6 alkyl and wherein R3 is SR6 or SO2R6, wherein R6 is selected from the group consisting of H, C1-C6 alkyl, aminoalkyl, pyrrolidinoethyl, piperidinoethyl, dimethylaminoethyl and diethylaminoethyl, and a pharmaceutically acceptable carrier, inorganic salt, diluent, glidant, lubricant, excipient, sweetening agent, wetting agent, absorbent and/or retardant therefor.

A mercaptophenyl maphthyl methane compound having the structural formula 1:

• wherein R is CHOH, wherein R1 is H or C1-C6 alkyl, wherein R2 is H or C1-C6 alkyl, and wherein R3 is SR6 wherein R6 is C1-C6 alkyl.

A pharmaceutical composition comprising a mercaptophenyl naphthyl methane compound having the structural formula 1:

• wherein R is CHOH, wherein R1 is H or C1-C6 alkyl, wherein R2 is H or C1-C6 alkyl, and wherein R3 is SR6 wherein R6 is C1-C6 and a pharmaceutically acceptable carrier, inorganic salt, diluent, glidant, lubricant, excipient, sweetening agent, wetting agent, absorbent and/or retardant therefor alkyl.