US 7,115,613 B2 · Selected fused pyrrolocarbazoles

Abstract

The present invention relates generally to selected fused pyrrolocarbazoles, including pharmaceutical compositions thereof and methods of treating diseases therewith. The present invention is also directed to intermediates and processes for making these fused pyrrolocarbazoles.

Claims8

Dependent claims

Compounds of Formula I:

wherein R1 and R3 are in accordance with the following table:
Cmpd
R1
R3
27
CH2CH2CH2OH
CH2SCH(CH3)2
37
CH2CH2CH2OCOCF3
CH2SCH2CH2CH3
39
CH2CH2CH2OH
CH2S(2-pyrimidyl).

10 more elements

Dependencies are inferred from the claim text.

Facts

Application

10/400,136Filed 26 Mar 2003 · continuation

Priority

25 Aug 2000

Published

US 2003/0203957 A130 Oct 2003

Granted

3 Oct 2006

Term ends

Not estimatedThe source records don’t support an estimate.

Classification33 codes

C07D 487/04
In which the condensed system contains two hetero rings: ortho-condensed systems
A61K 31/407
Having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil: condensed with other…
A61P 3/00
Drugs for disorders of the metabolism
A61P 3/10
For glucose homeostasis: for hyperglycaemia, e.g. antidiabetics

Family

Application60/227,803Us provisional application · filed 25 Aug 2000

Application60/278,455Us provisional application · filed 23 Mar 2001

Application09/935,285Parent of this continuation · filed 22 Aug 2001

US 2003/0203957 A1Pre-grant publication · published 30 Oct 2003

US 6,630,500 B2Parent of this continuation

US 2002/0061920 A1Published application

US 7,115,613 B2This patent

From the US filing history. Foreign family members aren’t listed.

Abstract

Facts

Application

10/400,136Filed 26 Mar 2003 · continuation

Priority

25 Aug 2000

Published

US 2003/0203957 A130 Oct 2003

Granted

3 Oct 2006

Term ends

Not estimatedThe source records don’t support an estimate.

Classification33 codes

C07D 487/04
In which the condensed system contains two hetero rings: ortho-condensed systems
A61K 31/407
Having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil: condensed with other…
A61P 3/00
Drugs for disorders of the metabolism
A61P 3/10
For glucose homeostasis: for hyperglycaemia, e.g. antidiabetics

Family

Application60/227,803Us provisional application · filed 25 Aug 2000

Application60/278,455Us provisional application · filed 23 Mar 2001

Application09/935,285Parent of this continuation · filed 22 Aug 2001

US 2003/0203957 A1Pre-grant publication · published 30 Oct 2003

US 6,630,500 B2Parent of this continuation

US 2002/0061920 A1Published application

US 7,115,613 B2This patent

From the US filing history. Foreign family members aren’t listed.

Selected fused pyrrolocarbazoles

Life of this patent

Abstract

Claims8

Selected fused pyrrolocarbazoles

Life of this patent

Abstract

Claims8