Fused bicyclic pyridine derivatives as tachykinin receptor antagonists
AssigneeKyorin Pharmaceutical.Co., Ltd.
InventorsShigeki Seto, Asao Tanioka, Makoto Ikeda, Shigeru Izawa
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AssigneeKyorin Pharmaceutical.Co., Ltd.
InventorsShigeki Seto, Asao Tanioka, Makoto Ikeda, Shigeru Izawa
Estimating the term…
A novel fused bicyclic pyridine derivative or a salt thereof that acts as a tachykinin receptor antagonist, in particular as an NK1 receptor antagonist, is represented by the following general formula (1): wherein the rings A and B are each a benzene ring which may have 1 to 3 substituents (any adjacent two of which may be bound to one another to form a ring); the ring C is a nitrogen-containing ring having a hydrogen atom substituted with a nitrogen atom; R1 and R2 are each independently a hydrogen atom, a C1 to C6 alkyl group, a C1 to C6 alkylsulfonyl group, a C1 to C6 alkylcarbonyl group, or a C1 to C6 alkoxycarbonyl group, or R1 and R2 are bound to one another to form the ring D; m is 1 or 2; n is 2 or 3; and q is an integer from 1 to 4.
A compound of formula (1), or a salt thereof:
A compound of formula (1a), or a salt thereof:
Dependencies are inferred from the claim text.