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US 6,617,460 B1Granted
Process for preparing toluenesulfinates
AssigneeEli Lilly and Company
InventorsBenjamin Alan Anderson, Nancy Kay Harn, Richard Duane Miller, Edward Francis Plocharczyk
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Abstract
A process for preparing novel compounds useful in the preparation of 1H-indole-3-glyoxamides.
Claims3
An intermediate compound of the formula V1
- wherein:
- R is selected from the group consisting of —(C1-C6)alkyl, aryl and substituted aryl
- R2 is selected from the group consisting of C7-C20 alkyl;
- where;
- R10 is selected from the group consisting of halo, C1-C10 alkyl, C1-C10 alkoxy, —S—(C1-C10 alkyl) and halo (C1-C10)alkyl, and t is an integer from 0 to 5 both inclusive;
- R2 is [selected from the group consisting of hydrogen, halo, C1-C3 alkyl, C3-C4 cycloalkyl, C3-C4 cycloalkenyl, —O—(C1-C2 alkyl), —S—(C1-C2 alkyl), aryl, aryloxy, and HET;] a heterocyclic group selected from the group consisting of thiazole, isothiazole, oxadiazole, and imidazole;
- R5 is selected from the group consisting of hydrogen, (C1-C6)alkyl, (C1-C6)alkoxy, halo(C1-C6)alkoxy, halo(C2-C6)alkyl, bromo, chloro, fluoro, iodo and aryl.
4 more elements
Dependencies are inferred from the claim text.