Fluorinated imidazoline benzodioxane, preparation and therapeutic uses thereof
AssigneePierre Fabre Medicament
InventorsThierry Imbert, Patrice Mayer, Marc Marien, Peters Pauwels
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Abstract
The present invention relates to novel fluorinated benzodioxane imidazoline derivatives, to their preparation and to their therapeutic applications. The invention is directed more particularly toward the compounds corresponding to the structure of general formula 1: in which: R represents a linear, branched or cyclized alkyl or alkenyl group containing 1 to 7 carbon atoms, or a benzyl group, and the fluorine atom can occupy position 5, 6, 7 or 8, in their racemic form and their dextrorotatory and levorotatory pure enantiomeric forms, and also the addition salts thereof.
Claims19
A compound corresponding to the structure of general formula 1:
- in which:
- R represents a linear, branched or cyclized alkyl or alkenyl group containing 1 to 7 carbon atoms, or a benzyl group, and
- the fluorine atom can occupy position 5, 6, 7 or 8, in their racemic form and their dextrorotatory and levorotatory pure enantiomeric forms, and also the addition salts thereof.
Dependencies are inferred from the claim text.