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US 6,548,449 B1Granted
Substituted phenyluracils with herbicidal effect
AssigneeBayer Aktiengesellschaft
InventorsRoland Andree, Markus Dollinger, Mark Wilhelm Drewes, Ingo Wetcholowsky, Randy Allen Myers
Life of this patent
Estimating the term…
Abstract
The invention relates to novel substituted phenyluraciles of the general formula (I) in which m, n, Q and R1-7 are each as defined in the description, and to processes for their preparation and to their use as herbicides.
Claims11
A phenyluracil of the formula (I)
- in which
- m represents the numbers 0, 1 or 2,
- n represents the numbers 0, 1, 2 or 3,
- Q represents O, S, SO, SO2, NH or N(C1-C4-alkyl),
- R1 represents hydrogen, amino or optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl having 1 to 6 carbon atoms,
- R2 represents carboxyl, cyano, carbamoyl, thiocarbamoyl, or represents in each case optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl or alkoxy-carbonyl having in each case up to 6 carbon atoms,
- R3 represents hydrogen, halogen or optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl having 1 to 6 carbon atoms,
- R4 represents hydrogen, cyano or halogen,
- R5 represents nitro, amino, hydroxyl, carboxyl, cyano, carbamoyl, thiocarbamoyl, sulpho, chlorosulphonyl, aminosulphonyl, halogen, or represents in each case optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl, alkoxy, alkyl-thio, alkylsulphinyl, alkylsulphonyl, alkylamino, alkylcarbonyl, alkoxycarbonyl, alkylaminocarbonyl, alkylcarbonylamino, alkoxycarbonylamino or alkyl-sulphonylamino having in each case up to 6 carbon atoms, and
- R6 represents amino or one of the groupings below —NH—R8, —N(R8)2, —NH—SO2—R8, —N(R8)(SO2—R8), —N(SO2—R8)2, —NH—CO—R9, —N(R8)(CO—R9), —N(CO—R9)2, —N(SO2—R8)(CO—R9),
- R7 represents nitro, amino, hydroxyl, mercapto, carboxyl, cyano, carbamoyl, thio-carbamoyl, sulpho, chlorosulphonyl, aminosulphonyl, halogen, or represents in each case optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino, alkylcarbonyl, alkoxycarbonyl, alkylaminocarbonyl, alkylcarbonylamino, alkoxycarbonyl-amino, alkylsulphonylamino or bis-alkylsulphonyl-amino having in each case up to 6 carbon atoms,
- R8 represents optionally halogen-substituted alkyl having 1 to 6 carbon atoms, represents optionally halogen-substituted alkenyl having 2 to 6 carbon atoms, represents optionally cyano-, halogen- or C1-C4-alkyl-substituted cycloalkyl having 3 to 6 carbon atoms, represents in each case optionally nitro-, cyano-, thiocarbamoyl-, halogen-, C1-C4-alkyl, C1-C4-halogenoalkyl-, C1-C4-alkoxy-, C1-C4-halogenoalkoxy-, C1-C4-alkylthio-, C1-C4-halogenoalkylthio-, C1-C4-alkylsulphinyl-, C1-C4-halogenoalkylsulphinyl-, C1-C4-alkylsulphonyl-, C1-C4-halogenoalkylsulphonyl- or C1-C4-alkoxy-carbonyl-substituted aryl or arylalkyl having in each case 6 or 10 carbon atoms in the aryl group and optionally 1 to 4 carbon atoms in the alkyl moiety, or represents optionally cyano-, halogen-, C1-C4-alkyl-, C1-C4-halogenoalkyl-, C1-C4-alkoxy-, C1-C4-halogenoalkoxy-, C1-C4-alkylthio-, C1-C4-halogenoalkylthio-, C1-C4-alkylsulphinyl-, C1-C4-halogenoalkylsulphinyl-, C1-C4-alkylsulphonyl- or C1-C4-halogenoalkyl-sulphonyl-substituted heterocyclyl selected from the group consisting of furyl, thienyl, oxazolyl, isoxazolyl, pyrazolyl, pyridyl and pyrimidyl, and
- R9 represents hydrogen, represents in each case optionally cyano-, halogen- or C1-C4-alkoxy-substituted alkyl, alkoxy, alkylamino or dialkylamino having in each case 1 to 6 carbon atoms, represents in each case optionally cyano- or halogen-substituted alkenyl or alkinyl having in each case 2 to 6 carbon atoms, represents in each case optionally cyano-, halogen- or C1-C4-alkyl-substituted cycloalkyl or cycloalkylalkyl having in each case 3 to 6 carbon atoms in the cycloalkyl group and optionally 1 to 4 carbon atoms in the alkyl moiety, represents in each case optionally nitro-, cyano-, thiocarbamoyl-, halogen-, C1-C4-alkyl-, C1-C4-halogenoalkyl-, C1-C4-alkoxy-, C1-C4-halogenoalkoxy-, C1-C4-alkylthio-, C1-C4-halogenoalkylthio-, C1-C4-alkylsulphinyl-, C1-C4-halogenoalkylsulphinyl-, C1-C4-alkylsulphonyl-, C1-C4-halogenoalkylsulphonyl- or C1-C4-alkoxy-carbonyl-substituted aryl or arylalkyl having in each case 6 or 10 carbon atoms in the aryl group and optionally 1 to 4 carbon atoms in the alkyl moiety, or represents optionally cyano-, halogen-, C1-C4-alkyl-, C1-C4-halogenoalkyl-, C1-C4-alkoxy-, C1-C4-halogenoalkoxy-, C1-C4-alkylthio-, C1-C4-halogenoalkylthio-, C1-C4-alkylsulphinyl-, C1-C4-halogenoalkylsulphinyl-, C1-C4-alkylsulphonyl- or C1-C4-halogenoalkyl-sulphonylsubstituted heterocyclyl selected from the group consisting of furyl, thienyl, oxazolyl, isoxazolyl, pyrazolyl, pyridyl and pyrimidyl.
10 more elements
A phenyluracil of the formula (I)
- wherein
- m represents the number 0,
- n represents the number 1,
- Q represents 0,
- R1 represents methyl,
- R2 represents trifluoromethyl,
- R3 represents hydrogen,
- R4 represents fluorine or chlorine,
- R6 represents, amino, —NH—SO2—R8 or —N(SO2—R8)(CO—R9),
- R7 represents nitro, cyano, fluorine, chlorine, bromine or represents optionally fluorine-substituted methyl or methoxy,
- R8 represents methyl or ethyl, and
8 more elements
Dependencies are inferred from the claim text.