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US 6,444,616 B1Granted
Substituted p-trifluoromethylphenyluracils
AssigneeBayer Aktiengesellschaft
InventorsMark-Wilhelm Drewes, Roland Andree, Markus Dollinger
Life of this patent
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Abstract
The invention relates to novel substituted p-trifluoromethylphenyluracils of the general formula (I) in which R1, R2, R3, R4 and R5 are each as defined in the description, to a process for their preparation and to their use as herbicides.
Claims4
A substituted p-trifluoromethylphenyluracil of the formula (I)
- wherein
- R1 represents hydrogen, cyano, fluorine, chlorine or bromine,
- R2 represents a grouping A1—A2—A3 wherein
- A1 represents a single bond, O, S, —SO—, or
- A1 represents C1-C6-alkanediyl, C2-C6-alkenediyl, C2-C6-alkynediyl, C3-C6-cycloalkanediyl, C3-C6-cycloalkenediyl or phenylene, each of which is optionally substituted by fluorine or chlorine,
- A2 represents a single bond, represents O, S, —SO—, —SO2—, —CO— or the grouping
- in which A4 represents hydrogen, hydroxyl, C1-C4-alkyl, C1-C4-alkoxy, phenyl, C1-C4-alkylsulphonyl or phenylsulphonyl, or
- A2 represents C1-C6-alkanediyl, C2-C6-alkenediyl, C2-C6-alkynediyl, C3-C6-cycloalkanediyl, C3-C6-cycloalkenediyl or phenylene, each of which is unsubstituted or substituted by fluorine or chlorine,
- A3 represents hydrogen, hydroxyl, mercapto, amino, cyano, isocyanato, thiocyanato, nitro, carboxyl, carbamoyl, thiocarbamoyl, sulpho, chlorosulphonyl, halogen;
- represents alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino, dialkylamino, alkoxycarbonyl or dialkoxy(thio)phosphoryl having in each case 1 to 6 carbon atoms in the alkyl groups and being in each case unsubstituted or substituted by fluorine, chlorine, bromine or C1-C4-alkoxy;
- represents alkenyl, alkenyloxy, alkenylamino, alkylideneamino, alkenyloxycarbonyl, alkynyl, alkynyloxy, alkynylamino or alkynyloxycarbonyl having in each case 2 to 6 carbon atoms in the alkenyl, alkylidene or alkynyl groups and being in each case unsubstituted or substituted by fluorine, chlorine or bromine;
- represents cycloalkyl, cycloalkyloxy, cycloalkylalkyl, cycloalkylalkoxy, cycloalkylideneamino, cycloalkyloxycarbonyl or cycloalkylalkoxycarbonyl having in each case 3 to 6 carbon atoms in the cycloalkyl groups and 0 to 4 carbon atoms in the alkyl groups and being in each case unsubstituted or substituted by a moiety selected from the group consisting of fluorine, chlorine, bromine, cyano, carboxyl, C1-C4-alkyl and C1-C4-alkoxy-carbonyl;
- represents phenyl, phenyloxy, phenyl-C1-C4-alkyl, phenyl-C1-C4-alkoxy, phenyloxycarbonyl or phenyl-C1-C4-alkoxy-carbonyl, each of which is unsubstituted or substituted by a moiety selected from the group consisting of nitro, cyano, carboxyl, fluorine, chlorine, bromine, C1-C4-alkyl, C1-C4-halogenoalkyl, C1-C4-alkyloxy, C1-C4-halogenoalkyloxy and C1-C4-alkoxycarbonyl;
- or
- represents in each case unhydrogenated or fully or partially hydrogenated pyrrolyl, pyrazolyl, imidazolyl, triazolyl, furyl, thienyl, oxazolyl, isoxazolyl, thiazolyl, isothiazolyl, oxadiazolyl, thiadiazolyl, pyridinyl, pyrimidinyl, triazinyl, pyrazolyl-C1-C4-alkyl, furyl-C1-C4-alkyl, thienyl-C1-C4-alkyl, oxazolyl-C1-C4-alkyl, isoxazol-C1-C4-alkyl, thiazole-C1-C4-alkyl, pyridinyl-C1-C4-alkyl, pyrimidinyl-C1-C4-alkyl, pyrazolylmethoxy, furylmethoxy, perhydropyranylmethoxy or pyridylmethoxy,
- R3 represents hydrogen, fluorine, chlorine, bromine or unsubstituted or fluorine or chlorine-substituted or fluorine- and chlorine-substituted alkyl having 1 to 4 carbon atoms,
- R4 represents unsubstituted or fluorine- or chlorine-substituted or fluorine- and chlorine-substituted alkyl having 1 to 4 carbon atoms, and
- R5 represents amino.
15 more elements
Dependencies are inferred from the claim text.