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US 6,310,005 B1Granted
Isothiazole carboxylic acid amides
AssigneeBayer Aktiengesellschaft
InventorsLutz Assmann, Hans-Ludwig Elbe, Dietmar Kuhnt, Gerd Hänssler, Karl-Heinz Kuck, Yoshinori Kitagawa, Haruko Sawada, Haruhiko Sakuma
Life of this patent
Estimating the term…
Abstract
Novel isothiazolecarboxamides of the formula in which R is as defined in the description, a plurality of processes for preparing the novel compounds and their use for protecting plants against attack by undesirable microorganisms.
Claims9
An isothiazolecarboxamide of the formula
- wherein
- R represents a radical of the formula
- —A1—R5,
- wherein
- A1 represents —CH2—, —CH2—CH2— or
- and
- R5 represents thiazolidinethion-3-yl, morpholinyl, piperazinyl, pyrazolyl, imidazolyl, 1,2,4-triazolyl, pyrrolyl, thienyl, thiazolyl, isothiazolyl, oxazolyl, isoxazolyl, pyridinyl, pyrimidinyl, triazinyl, 1,2,3-triazolyl, benzotriazolyl, quinolinyl, isoquinolinyl, quinazolinyl, indolyl, benzothienyl, benzofuranyl, benzothiazolyl or benzimidazolyl, where these radicals may be unsubstituted or mono- or disubstituted by identical or different substituents from the group consisting of fluorine, chlorine, bromine, cyano, nitro, carboxyl, methyl, ethyl, propyl, isopropyl, n-butyl, sec-butyl, iso-butyl, tert-butyl, halogenoalkyl having 1 or 2 carbon atoms and 1 to 3 fluorine, chlorine and/or bromine atoms, methoxycarbonyl, ethoxycarbonyl, methoxy, ethoxy, propoxy, isopropoxy, tert-butoxy, halogenoalkoxy having 1 or 2 carbon atoms and 1 to 3 fluorine, chlorine and/or bromine atoms, methylthio, ethylthio, halogenoalkylthio having 1 or 2 carbon atoms and 1 to 3 fluorine, chlorine and/or bromine atoms, methylamino, ethylamino, dimethylamino, diethylamino, phenyl and phenoxy, or
- R represents a radical of the formula
- wherein
- R1 represents hydrogen or alkyl having 1 to 4 carbon atoms,
- R2 represents alkoxy having 1 to 4 carbon atoms or represents morpholinyl, piperazinyl, pyrazolyl, imidazolyl, 1,2,4-triazolyl, pyrrolyl, thienyl, thiazolyl, isothiazolyl, oxazolyl, isoxazolyl, pyridinyl, pyrimidinyl, triazinyl or 1,2,3-triazolyl, where these radicals may be unsubstituted or mono- or disubstituted by identical or different substituents from the group consisting of fluorine, chlorine, bromine, cyano, nitro, carboxyl, methyl, ethyl, propyl, isopropyl, n-butyl, sec-butyl, iso-butyl, tert-butyl, halogenoalkyl having 1 or 2 carbon atoms and 1 to 3 fluorine, chlorine and/or bromine atoms, methoxycarbonyl, ethoxycarbonyl, methoxy, ethoxy, propoxy, isopropoxy, tert-butoxy, halogenoalkoxy having 1 or 2 carbon atoms and 1 to 3 fluorine, chlorine and/or bromine atoms, methylthio, ethylthio, halogenoalkylthio having 1 or 2 carbon atoms and 1 to 3 fluorine, chlorine and/or bromine atoms, methylamino, ethylamino, dimethylamino, diethylamino, phenyl and phenoxy, and
- m represents 1 or 2, or
- R represents a radical of the formula
- wherein
- R3 represents a heterocycle of the formula
- or represents morpholinyl, piperazinyl, pyrazolyl, imidazolyl, 1,2,4-triazolyl, pyrrolyl, thienyl, thiazolyl, isothiazolyl, oxazolyl, isoxazolyl, pyridinyl, pyrimidinyl, triazinyl or 1,2,3-triazolyl, where these radicals may be unsubstituted or mono- or disubstituted by identical or different substituents from the group consisting of fluorine, chlorine, bromine, cyano, nitro, carboxyl, methyl, ethyl, propyl, isopropyl, n-butyl, sec-butyl, iso-butyl, tert-butyl, halogenoalkyl having 1 or 2 carbon atoms and 1 to 3 fluorine, chlorine and/or bromine atoms, methoxycarbonyl, ethoxycarbonyl, methoxy, ethoxy, propoxy, isopropoxy, tert-butoxy, halogenoalkoxy having 1 or 2 carbon atoms and 1 to 3 fluorine, chlorine and/or bromine atoms, methylthio, ethylthio, halogenoalkylthio having 1 or 2 carbon atoms and 1 to 3 fluorine, chlorine and/or bromine atoms, methylamino, ethylamino, dimethylamino, diethylamino, phenyl and phenoxy or
- R3 represents a radical of the formula
- wherein
- R4 represents cyclopropyl, cyclopentyl or cyclohexyl, and
- n represents 1 or 2, or
- R represents morpholinyl, piperazinyl, pyrazolyl, imidazolyl, 1,2,4-triazolyl, pyrrolyl, thienyl, thiazolyl, isothiazolyl, oxazolyl, isoxazolyl, pyridinyl, pyrimidinyl, triazinyl, 1,2,3-triazolyl, benzotriazolyl, quinolinyl, isoquinolinyl, quinazolinyl, indolyl, benzothienyl, benzofuranyl, benzothiazolyl or benzimidazolyl, where these radicals may be unsubstituted or mono- or disubstituted by identical or different substituents from the group consisting of fluorine, chlorine, bromine, cyano, nitro, carboxyl, methyl, ethyl, trifluoromethyl, difluoromethyl, trichloromethyl, methoxycarbonyl, ethoxycarbonyl, methoxy, ethoxy, trifluoromethoxy, methylthio, trifluoromethylthio, methylamino, dimethylamino, phenyl and phenoxy.
18 more elements
Dependencies are inferred from the claim text.