N-heterocyclic methylpropylamine derivatives, process for producing the same and germicides
AssigneeKureha Kagaku Kogyo Kabushiki Kaisha
InventorsAtsushi Ito, Satoru Kumazawa, Keiichi Sudo, Tsumoru Watanabe, Takayoshi Eizuka, Yoshitaka Niizeki
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Abstract
N-heterocyclicmethylpropylamine derivatives of formula (I): and acid addition salts thereof; wherein R1 represents hydrogen, halogen, alkyl, alkenyl, halogenated alkyl, alkoxy, halogenated alkoxy, hydroxyl, cyano, nitro, phenyl optionally having a substituent on a ring thereof or phenoxy; n represents an integer of 0-5; R2 represents a heterocycle containing at least one nitrogen atom as the hetero atom and optionally having a substituent on a ring thereof; and R3 represents hydrogen or C1-C5 alkyl.
Claims2
An N-heterocyclicmethylpropylamine derivative of formula (I):
- or an acid addition salt thereof;
- wherein R1 represents a moiety selected from the group consisting of hydrogen, halogen, C1-C6 alkyl, C1-C6 alkenyl, C1-C6 halogenated alkyl, C1-C6 alkoxy, C1-C6 halogenated alkoxy, hydroxyl, cyano, nitro, phenyl optionnally having a substituent on a ring thereof and phenoxy;
- n represents an integer of 0-5;
- when n is 2 or greater, each R1 may be the same or different and two R1 groups may be bonded together to form a ring selected from a group consisting of indane, 1,2-methylenedioxybenzene and naphthalene;
- R2 represents a heterocycle selected from a group consisting of pyridine, pyrazine, pyrimidine, thiazole, oxazole, pyrazole and pyrrole, said heterocycle optionally having a substituent on a ring thereof;
- and R3 represents a moiety selected from the group consisting of hydrogen and C1-C5 alkyl,
- with the proviso that the following compounds are excluded:
- N-[3-(4-t-butylphenyl)-2-methylpropyl]-N-(t-butyl)-3-pyridylmethylamine,
- N-[3-(4-t-butylphenyl)-2-methylpropyl]-N-butyl-3-pyridylmethylamine, and
- N-[3-(4-t-butylphenyl)-2-methylpropyl]-N-methyl-3-pyridylmethylamine.
A fungicide compound containing as an effective ingredient, an N-heterocyclicmethylpropylamine derivative of formula (I):
- or an acid addition salt thereof;
- wherein R1 represents a moiety selected from the group consisting of hydrogen, halogen, C1-C6 alkyl, C1-C6 alkenyl, C1-C6 halogenated alkyl, C1-C6 alkoxy, C1-C6 halogenated alkoxy, hydroxyl, cyano, nitro, phenyl optionally having a substituent on a ring thereof and phenoxy;
- n represents an integer of 0-5;
- when n is 2 or greater, each R1 may be the same or different and two R1 groups may be bonded together to form a ring selected from a group consisting of indane, 1,2-methylenedioxybenzene and naphthalene;
- R2 represents a heterocycle selected from a group consisting of pyridine, pyrazine, pyrimidine, thiazole, oxazole, pyrazole and pyrrole, said heterocycle optionally having a substituent on a thereof;
- and R3 represents a moiety selected from the group consisting of hydrogen and C1-C5 alkyl,
- with the proviso that the following compounds are excluded:
- N-[3-(4-t-butylphenyl)-2-methylpropyl]-N-(t-butyl)-3-pyridylmethylamine,
- N-[3-(4-t-butylphenyl)-2-methylpropyl]-N-butyl-3-pyridylmethylamine, and
- N-[3-(4-t-butylphenyl)-2-methylpropyl]-N-methyl-3-pyridylmethylamine.
Dependencies are inferred from the claim text.