4-jod-2[N-(N-alkyl-aminocarbonyl)-aminosulfonyl]-benzoic acid methyl ester and derivatived thereof and method for their production
AssigneeHoechst Schering AgrEvo GmbH
InventorsLothar Willms, Harald Knorr
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AssigneeHoechst Schering AgrEvo GmbH
InventorsLothar Willms, Harald Knorr
Estimating the term…
The invention relates to compounds of the formula (I) ##STR1## in which R=(subst.) alkyl or (subst.) cycloalkyl, which are suitable as intermediates for preparing herbicidal sulfonylureas. According to the invention, the compounds (I) are prepared by (a) diazotizing a compound of the formula (II) ##STR2## in the presence of an acid H.sup.+ X.sup.-, where X.sup.- is an equivalent of an anion, to give the novel compounds (diazonium salts) of the formula (III) ##STR3## (b) reacting the compound of the formula (III) in the presence of iodide ions to give the compound (IV) and ##STR4## (c) reacting the compound of the formula (IV) with an isocyanate of the formula (V) R--N.dbd.C.dbd.O (V) in which R is as defined in formula (I), to give the compound of the formula (I).
A compound of the formula (I), ##STR10## in which R is alkyl or cycloalkyl, each of the last two radicals being unsubstituted or substituted.
A process for preparing compounds of the formula ##STR11## in which R is alkyl or cycloalkyl, each of the last two radicals being unsubstituted or substituted
A process for preparing a compound of the formula ##STR15## in which R is alkyl or cycloalkyl, each of the last two radicals being unsubstituted or substituted,
Dependencies are inferred from the claim text.