Use of 4-phenyl-3,6-dihydro-2H-pyridyl derivatives
AssigneeHoffmann-La Roche Inc.
InventorsAnne Bourson, Gunther Fischer, Marie-Paule Heitz Neidhart, Vincent Mutel, Gerhard Trube
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AssigneeHoffmann-La Roche Inc.
InventorsAnne Bourson, Gunther Fischer, Marie-Paule Heitz Neidhart, Vincent Mutel, Gerhard Trube
Estimating the term…
The present invention relates to the use of compounds of general formula ##STR1## wherein R.sup.1 is hydrogen, halogen, lower alkyl or lower alkoxy; R.sup.2 is hydrogen; R.sup.3 is hydrogen, amino, ureido, lower alkylcarbonyl, lower alkyl-sulfonylamino, lower alkylcarbamoyl, carbamoyl, lower alkyloxycarbamoyl, lower alkylamino or R.sup.2 and R.sup.3 taken together are --(CH.sub.2).sub.m -- X is methylene, hydroxymethylene, lower alkoxymethylene or carbonyl, n is 0, 1 or 2 and m is 3 or 4 as well as pharmaceutically acceptable salts for the control or treatment of diseases which represent therapeutic indications for NMDA receptor subtype specific blockers.
A method for the control or treatment of diseases caused by over activation of NMDA receptor subtypes comprising orally administering to a host in need of such control or treatment, a compound of the formula ##STR8## wherein R.sup.1 is hydrogen, halogen, lower alkyl or lower alkoxy;
A method for the control or treatment of diseases caused by over activation of NMDA receptor subtypes comprising administering to a host in need of such control or treatment, a compound of the formula ##STR9## wherein R.sup.1 is hydrogen, halogen, lower alkyl or lower alkoxy;
Dependencies are inferred from the claim text.