Back to results
US 5,795,914 AGranted
Phenylalkan(en)oic acid
AssigneeOno Pharmaceutical Co., Ltd.
InventorsMitoshi Konno, Takahiko Nakae, Nobuyuki Hamanaka
Life of this patent
Estimating the term…
Abstract
The phenylalkan(en)oic acids of the formula: ##STR1## wherein the substituents are defined in the specification.
Claims3
A phenylkan(en)oic acid of the formula:
- ##STR191## wherein A is:
- --O--;
- W is:
- i) C.sub.1-13 alkylene,
- ii) phenylene, or ##STR192## R.sup.1 is:
- i) hydrogen,
- ii) C.sub.1-4 alkyl,
- iii) --COOH,
- iv) ##STR193## or v) --CH.sub.2 OH;
- two R.sup.2 are the same or different,
- i) hydrogen or
- ii) C.sub.1-4 alkyl;
- Y is ethylene or vinylene;
- D is:
- i) --Z--B, or ##STR194## Z is C.sub.3-11 alkylene or alkenylene;
- B is ##STR195## R.sup.3 is:
- i) hydrogen,
- ii) halogen,
- iii) C.sub.1-8 alkyl, alkoxy or alkylthio, or
- iv) C.sub.2-8 alkenyl, alkenyloxy or alkenylthio;
- n is 1-3;
- R.sup.4 is C.sub.1-7 alkylene;
- R.sup.5 is:
- i) C.sub.1-12 alkyl,
- ii) C.sub.2-12 alkenyl,
- iii) C.sub.5-7 cycloalkyl, or
- iv) phenethyl or phenethyl wherein the ring is substituted by one C.sub.1-4 alkoxy;
- with the proviso that:
- i) --A--W--R.sup.1 should bind to the 3- or 4-carbon in the benzene ring, and
- ii) when W is phenylene or ##STR196## A does not represent --O--;
- and non-toxic salts thereof.
28 more elements
Dependencies are inferred from the claim text.