Anilide derivatives and their use for combating botrytis
AssigneeBASF SE
InventorsKarl Eicken, Norbert Goetz, Albrecht Harreus, Eberhard Ammermann, Gisela Lorenz, Harald Rang
Life of this patent
Estimating the term…
Abstract
The use of nicotinic anilide derivatives of the general formula ##STR1## where the substituents have the following meanings: R.sup.1 halogen, methyl, trifluoromethyl, methoxy, methylthio, methylsulfinyl, methylsulfonyl R.sup.2 unsubstituted or halogen-substituted alkyl, unsubstituted or halogen-substituted alkenyl, alkynyl, unsubstituted or halogen-substituted alkoxy, unsubstituted or halogen-substituted alkenyloxy, alkynyloxy, cycloalkyl, cycloalkenyl, cycloalkyloxy, cycloalkenyloxy for combating Botrytis, and nicotinic anilides of the formula I.
Claims11
A method for treating Botrytis infestation comprising applying to a subject in need thereof, an effective amount of a compound of formula ##STR36## wherein A has the following meaning:
- thiazol-5-yl substituted in the 2- and 4-positions by hydrogen, methyl, chlorine or trifluoromethyl;
- and
- R has the following meanings:
- unsubstituted C.sub.3 -C.sub.12 -alkyl, unsubstituted C.sub.3 -C.sub.12 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, unsubstituted C.sub.3 -C.sub.12 -alkenyloxy, C.sub.3 -C.sub.12 -alkynyloxy, unsubstituted or C.sub.1 -C.sub.4 -alkyl-substituted C.sub.3 -C.sub.6 -cycloalkyl, unsubstituted or C.sub.1 -C.sub.4 -alkyl-substituted C.sub.4 -C.sub.6 -cycloalkenyl, unsubstituted or C.sub.1 -C.sub.4 -alkyl substituted C.sub.5 -C.sub.6 -cycloalkyloxy, unsubstituted or C.sub.1 -C.sub.4 -alkyl substituted C.sub.5 -C.sub.6 -cycloalkenyloxy, or phenyl which is unsubstituted or substituted by C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.3 -C.sub.4 alkylthio or halogen;
- in a suitable carrier.
A method for treating Botrytis infestation comprising applying to a subject in need thereof, an effective amount of a 2-aminobiphenyl compound of formula III ##STR37## wherein A has the following meaning:
- ##STR38## R.sup.4 methyl, trifluoromethyl, or chlorine;
- R.sup.5 is hydrogen, methyl, or chlorine;
- and
- R.sup.8 is C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkylthio or halogen;
- in a suitable carrier.
A method for treating Botrytis infestation comprising applying to a subject in need thereof, an effective amount of a 2-aminobiphenyl compound of formula IV ##STR39## wherein A has the following meaning:
- ##STR40## wherein R.sup.4 and R.sup.5 are as follows:
- R.sup.4 is methyl and R.sup.5 is hydrogen;
- or R.sup.4 is methyl and R.sup.5 is chlorine;
- or R.sup.4 is trifluoromethyl and R.sup.5 is hydrogen;
- or R.sup. 4 is trifluoromethyl and R.sup.5 is methyl;
- or R.sup. 4 is trifluoromethyl and R.sup.5 is chlorine;
- or R.sup.4 is chlorine and R.sup.5 is hydrogen;
- or R.sup.4 is chlorine and R.sup.5 is methyl;
- or R.sup.4 is chlorine and R.sup.5 is chlorine;
- in a suitable carrier.
A method for treating Botrytis infestation comprising applying to a subject in need thereof, an effective amount of a carboxanilide compound of formula V ##STR41## wherein A has the following meaning:
- ##STR42## R.sup.3 is methyl, trifluoromethyl, or chlorine;
- R.sup.4 is hydrogen, methyl, or chlorine;
- and
- R.sup.7 is unsubstituted C.sub.3 -C.sub.12 -alkyl, unsubstituted C.sub.3 -C.sub.12 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, unsubstituted C.sub.3 -C.sub.12 -alkenyloxy, C.sub.3 -C.sub.12 -alkynyloxy, unsubstituted or C.sub.1 -C.sub.4 -alkyl-substituted C.sub.3 -C.sub.6 -cycloalkyl, unsubstituted or C.sub.1 -C.sub.4 -alkyl-substituted C.sub.4 -C.sub. 6-cycloalkenyl, unsubstituted or C.sub.1 -C.sub.4 -alkyl-substituted C.sub.5 -C.sub.6 -cycloalkyloxy, unsubstituted or C.sub.1 -C.sub.4 -alkyl substituted C.sub.5 -C.sub.6 -cycloalkenyloxy,
- in a suitable carrier.
Aminobiphenyl compounds of formula III ##STR43## wherein A has the following meaning:
- ##STR44## R.sup. 4 is methyl, trifluoromethyl, or chlorine;
- R.sup.5 is hydrogen, methyl, or chlorine;
- and
- R.sup.8 is C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy, C.sub.1 -C.sub.4 -alkylthio, halogen.
Aminobiphenyl compounds of formula IV ##STR45## wherein A has the following meaning:
- ##STR46## wherein R.sup.4 and R.sup.5 are as follows:
- R.sup.4 is methyl and R.sup.5 is hydrogen;
- or R.sup.4 is methyl and R.sup.5 is chlorine;
- or R.sup.4 is trifluoromethyl and R.sup.5 is hydrogen;
- or R.sup. 4 is trifluoromethyl and R.sup.5 is methyl;
- or R.sup.4 is trifluoromethyl and R.sup.5 is chlorine;
- or R.sup.4 is chlorine and R.sup.5 is hydrogen;
- or R.sup.4 is chlorine and R.sup.5 is methyl;
- or R.sup.4 is chlorine and R.sup.5 is chlorine.
Carboxanilide compounds of formula V ##STR47## wherein A has the following meaning:
- ##STR48## R.sup.3 is methyl, trifluoromethyl, or chlorine;
- R.sup.4 is hydrogen, methyl, or chlorine;
- and
- R.sup.7 is unsubstituted C.sub.3 -C.sub.12 -alkyl, unsubstituted C.sub.3 -C.sub.12 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, unsubstituted C.sub.3 -C.sub.12 -alkenyloxy, C.sub.3 -C.sub.12 -alkynyloxy, unsubstituted or C.sub.1 -C.sub.4 -alkyl-substituted C.sub.3 -C.sub.6 -cycloalkyl, unsubstituted or C.sub.1 -C.sub.4 -alkyl-substituted C.sub.4 -C.sub.6 -cycloalkenyl, unsubstituted or C.sub.1 -C.sub.4 -alkyl-substituted C.sub.5 -C.sub.6 -cycloalkyloxy, unsubstituted or C.sub.1 -C.sub.4 -alkyl-substituted C.sub.5 -C.sub.6 -cycloalkenyloxy, with the proviso that R.sup.7 is not 3-methyl-but-2-en-1-yl or 3-methyl-but-3-en-1-yl when R.sup.1 is trifluoromethyl.
A composition for treating Botrytis infestation comprising an effective amount of a compound of formula ##STR49## wherein A has the following meaning:
- thiazol-5-yl substituted in the 2- and 4-positions by hydrogen, methyl, chlorine or trifluoromethyl;
- and
- R has the following meanings:
- unsubstituted C.sub.3 -C.sub.12 -alkyl, unsubstituted C.sub.3 -C.sub.12 -alkenyl, C.sub.3 -C.sub.6 -alkynyl, unsubstituted C.sub.3 -C.sub.12 -alkenyloxy, C.sub.3 -C.sub.12 -alkynyloxy, unsubstituted or C.sub.1 -C.sub.4 -alkyl-substituted C.sub.3 -C.sub.6 -cycloalkyl, unsubstituted or C.sub.1 -C.sub.4 -alkyl-substituted C.sub.4 -C.sub.6 -cycloalkenyl, unsubstituted or C.sub.1 -C.sub.4 -alkyl substituted C.sub.5 -C.sub.6 -cycloalkyloxy, unsubstituted or C.sub.1 -C.sub.4 -alkyl substituted C.sub.5 -C.sub.6 -cycloalkenyloxy, or phenyl which is substituted by C.sub.1 -C.sub.4 -alkyl, C.sub.4 -C.sub.6 -alkoxy, C.sub.1 -C.sub.4 -alkylthio or halogen;
- in a suitable carrier.
Dependencies are inferred from the claim text.