Back to results
US 5,440,052 AGranted
Compositions useful as a cannabinoid receptor probe
AssigneeUniversity of Connecticut
InventorsAlexandros Makriyannis, Guo Yan, Vasiliki Abadji
Life of this patent
Estimating the term…
Abstract
A composition of matter, comprising a cannabinol compound having the structure ##STR1## wherein, Q is --C(R.sup.1) (Y.sup.1)--(CH.sub.2).sub.n ----Z.sup.1 ; R.sup.1 is --H or --CH.sub.3 ; Y.sup.1 is --CH.sub.3 or Y.sup.2 ; Y.sup.2 is --N.sub.3 or --NCS; n is 4 or 6; Z.sup.1 is --H, when Y.sup.1 is Y.sup.2, or is Z.sup.2, when Y.sup.1 is --CH.sub.3 ; and Z.sup.2 is --N.sub.3 or --NCS. This composition has good binding affinity to the cannabinoid receptor and therefore, is useful as a receptor probe.
Claims3
A cannabinol compound having the following structure ##STR6## wherein:
- Q is --C(R.sup.1) (Y.sup.1)--(CH.sub.2).sub.n --Z.sup.1 ;
- R.sup.1 is --H or --CH.sub.3 ;
- Y.sup.1 is --CH.sub.3 or Y.sup.2 ;
- Y.sup.2 is --N.sub.3 or --NCS;
- n is 4 or 6;
- Z.sup.1 is --H, when Y.sup.1 is Y.sup.2, or is Z.sup.2, when Y.sup.1 is --CH.sub.3 ;
- and
- Z.sup.2 is --N.sub.3 or --NCS.
5 more elements
Dependencies are inferred from the claim text.