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US 5,314,879 AGranted
Silanyl oxypropylamines endowed with antifungal activity
AssigneeMinistero Delli `Universita` E Della Ricerca Scientifica E Tecnologica
InventorsGiovanni Camaggi, Lucio Filippini, Marilena Gusmeroli, Carlo Garavaglia, Luigi Mirenna
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Abstract
The invention relates to the manufacture and use of aryl-propyl-aminic compounds having the following formula ##STR1## that have a high antifungal activity and are useful in the agricultural field as fungicides.
Claims9
Antifungal compounds useful in the agricultural field having the formula:
- ##STR7## wherein:
- R.sub.1 and R.sub.2, which may be either equal to, or different from, each other, represent H atoms, either linear or branched (C.sub.1 -C.sub.6)-alkyl groups,
- Ar-B groups in which Ar is a (C.sub.6, C.sub.10)-aryl or (C.sub.6, C.sub.10)-halo-aryl group and
- B is a (C.sub.1 -C.sub.4)-alkylene or (C.sub.1 -C.sub.2)-alkyl-(C.sub.1 -C.sub.4)-alkylene group,
- or R.sub.1 and R.sub.2 taken together with the N atom form a (C.sub.3 -C.sub.8)-heterocyclic group or a (C.sub.2 -C.sub.7)-heterocyclic group containing a second heteroatom selected from among O and S, said heterocyclic groups being optionally substituted with one or more C.sub.1 -C.sub.4 alkyl groups, (C.sub.6 -C.sub.10)-aryl groups, halogens, or Ar-B groups in which the symbols Ar and B have the same meanings are defined above;
- R.sub.3 represents a (C.sub.1 -C.sub.3)-alkyl group;
- R.sub.4 which, when m is greater than 1, may be either different from, or equal to, one another, represent halogen atoms, (C.sub.1 -C.sub.3)-alkyl groups or (C.sub.1 -C.sub.3)-halo-alkyl groups;
- m is an integer within the range of from 0 to 4;
- R', R", which may be either equal to, or different from, each other, represent H, (C.sub.1 -C.sub.3)-alkyl group or halogen atoms;
- n is an integer within the range of from 0 to 3;
- Y represents a ##STR8## group in which C, D, E, either equal to, or different from, one another, represent H atoms, (C.sub.1 -C.sub.4) alkyl groups, (C.sub.1 -C.sub.4)-haloalkyl groups, (C.sub.1 -C.sub.4) alkoxy groups, (C.sub.1 -C.sub.4)-halo-alkoxy groups, (C.sub.6,C.sub.10) -aryl groups, and (C.sub.6, C.sub.10)-haloaryl groups;
- their enantiomers and diastereoisomers and corresponding metal salts and complexes.
9 more elements
Dependencies are inferred from the claim text.