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US 5,290,784 AGranted
Aconitane derivatives used as a medication to treat addiction
AssigneeYueqian Qu
InventorsYueqian Qu, Peng Qu
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AssigneeYueqian Qu
InventorsYueqian Qu, Peng Qu
Estimating the term…
This invention relates to a medication to treat addicts who are addicted to drugs or narcotics (including opium, morphine, heroine, cocaine, marijuana, amphetamine, etc.), the preparative method of this medication, as well as the treatment method for the addicts by using this medication. This medication to treat addiction is aconitane deivative having structures of formula I or II, wherein the formula I, R=.alpha.--OCH.sub.3, .beta.--OCH.sub.3 or .alpha.--OH; R.sub.1 =OAcABz, OH, OABz or H; R.sub.2 =H or OH; R.sub.3 =H or OH; R.sub.4 =H or OH; R.sub.5 =H or OH; R.sub.6 =OCH.sub.3, OBz, OAc or OH; wherein the formula II, R.sub.1 =R.sub.2 =R.sub.3 =OH. This medication to treat addiction is characterized by no drug-dependence, high cure effect, fast action and low side effect. ##STR1##
A method to treat the withdrawal symptoms of narcotic addiction which comprises administering a withdrawal symptom effective amount of an aconitane derivative having the structures of formula I and II, inorganic acid salts therefore, or a mixture of two of the foregoing ##STR11## In formula I, R=.alpha.--OCH.sub.3, .alpha.--OH or .beta.--OCH.sub.3 ;
A method for the treatment of withdrawal symptoms of addiction to a drug selected from the group consisting of opium, morphine, heroin, cocaine, marijuana, and amphetamines which comprises administering a withdrawal symptom effective amount of an aconitane derivative having the structures of formula I and II, inorganic acid salts therefor, or a mixture of two of the foregoing ##STR12## wherein R=.alpha.--OCH.sub.3, .alpha.--OH, or .beta.--OCH.sub.3 ;
Dependencies are inferred from the claim text.