Azole derivatives
AssigneeImperial Chemical Industries PLC
InventorsPeter W. R. Caulkett, Geraint Jones, Michael G. Collis, Simon M. Poucher
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AssigneeImperial Chemical Industries PLC
InventorsPeter W. R. Caulkett, Geraint Jones, Michael G. Collis, Simon M. Poucher
Estimating the term…
A compound of the formula I ##STR1## wherein: R.sup.1 is hydrogen, (1-6C)alkyl, or (1-4C)alkanoyl; R.sup.2 is phenyl, a C-linked aromatic 5- or 6-membered heterocyclic ring containing one of oxygen and sulphur and/or one or two nitrogen, or (1-8C)alkyl, alkenyl or alkynyl unsubstituted or substituted by a phenyl or a C-linked aromatic 5- or 6-membered heterocylic ring containing one of oxygen and sulphur and/or one or two nitrogen, any phenyl being unsubstituted or substituted by one, two or three of (1-4C)alkyl, (1-4C)alkoxy, halogen, trifluoromethyl, hydroxy, benzyloxy and (1-5C)alkanoyloxy; A is N or CT in which T is hydrogen or (1-4C)alkyl; or a pharmaceutically acceptable salt thereof, processes for the manufacture of the compounds, and pharmaceutical compositions containing them. The compounds are useful as adenosine antagonists.
A compound of the formula I:
A compound of formula XII:
Dependencies are inferred from the claim text.