Pyrimidin-5-ylsulfonamides
AssigneeCiba-Geigy Corporation
InventorsBeat B/o/ hner, Werner F/o/ ry, Rolf Schurter, Georg Pissiotas
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AssigneeCiba-Geigy Corporation
InventorsBeat B/o/ hner, Werner F/o/ ry, Rolf Schurter, Georg Pissiotas
Estimating the term…
The invention relates to novel sulfonylureas of the formula I ##STR1## wherein R.sub.1 is hydrogen or C.sub.1 -C.sub.5 alkyl, R.sub.2 and R.sub.3, each independently of the other, are hydrogen, C.sub.1 -C.sub.5 alkyl, C.sub.1 -C.sub.5 alkoxy, C.sub.1 -C.sub.5 alkylthio, C.sub.1 -C.sub.5 haloalkyl, halogen, C.sub.1 -C.sub.5 haloalkylthio, C.sub.1 -C.sub.4 alkylamino, C.sub.1 -C.sub.4 dialkylamino, an alkoxyalkyl group or alkoxyalkoxy group, each containing not more than 6 carbon atoms, Z is oxygen or sulfur, E is --CH.dbd. or --N.dbd., and Q is an unsubstituted or substituted 6-membered heterocyclic radical containing 2 to 3 nitrogen atoms and bound through a carbon atom, and the salts thereof. A process for the preparation of the novel compounds and the use thereof are also described. The compounds of formula I can be used in the form of agriculturally useful compositions for controlling weeds and/or for selectively influencing plant growth.
A pyrimidin-5-sulfonamide of the formula ##STR50## wherein R.sup.a is hydrogen, halogen, C.sub.1-4 alkyl or C.sub.1 -C.sub.4 alkoxy, and
A compound according to claim 20, wherein R.sup.a is hydrogen, chlorine or methoxy and R.sup.b is chlorine, methoxy or trifluoromethyl.
Dependencies are inferred from the claim text.
From the US filing history. Foreign family members aren’t listed.
Heterocyclic compounds containing unspecified hetero rings
Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<: containing the group >N—CO—N< directly attached to at least one heterocyclic ring;…
With hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals,…:…
With hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals,…:…
Term ended 20 Dec 2005 (estimated)
USPTO file history isn’t available for this patent, so only indexed dates are shown.
The present invention relates to a group of novel sulfonylureas and sulfonylthioureas which have valuable growth regulating properties and which are suitable for selectively influencing plant growth, for the control of weeds e.g. in crops of useful plants and/or for influencing the phytotoxic properties of other herbicidal compounds. The invention also relates to the preparation of these sulfonylureas and sulfonylthioureas, and to agricultural compositions which contain them.
Accordingly, the invention relates to compounds of the formula I ##STR2## wherein
R.sub.1 is hydrogen or C.sub.1 -C.sub.5 alkyl,
In the following Examples parts and percentages are by weight.
The intermediates and final products listed in the following tables can be prepared in corresponding manner:
TABLE 1 ______________________________________ QSO.sub.2NH.sub.2 Abbre- Compound Q viation Physical data ______________________________________ 1.1 ##STR10## Q 1 m.p. 109-110.degree. C. 1.2 ##STR11## Q 2 m.p. 115-120.degree. C. 1.3 ##STR12## Q 3 1.4 ##STR13## Q 4 1.5 ##STR14## Q 5 1.6 ##STR15## Q 6 1.7 ##STR16## Q 7 1.8 ##STR17## Q 8 1.9 ##STR18## Q 9 1.10 ##STR19## Q 10 1.11 ##STR20## Q 11 1.12 ##STR21## Q 12 1.13 ##STR22## Q 13 1.14 ##STR23## Q 14 1.15 ##STR24## Q 15 1.16 ##STR25## Q 16 1.17 ##STR26## Q 17 1.18 ##STR27## Q 18 1.19 ##STR28## Q 19 1.20 ##STR29## Q 20 1.21 ##STR30## Q 21 1.22 ##STR31## Q 22 1.23 ##STR32## Q 23 1.24 ##STR33## Q 24 1.25 ##STR34## Q 25 1.26 ##STR35## Q 26 1.27 ##STR36## Q 27 1.28 ##STR37## Q 28 1.29 ##STR38## Q 29 1.30 ##STR39## Q 30 1.31 ##STR40## Q 31 1.32 ##STR41## Q 32 1.33 ##STR42## Q 33 1.34 ##STR43## Q 34 1.35 ##STR44## Q 35 1.36 ##STR45## Q 36 1.37 ##STR46## Q 37 1.38 ##STR47## Q 38 1.39 ##STR48## Q 39 ______________________________________