9-anthryloxyaminoalkanes and related compounds as anti-inflammatory and analgetic agents
AssigneeSyntex (U.S.A.) Inc.
InventorsPeter H. Nelson, Stefan H. Unger, Thomas R. Thieme
Life of this patent
Estimating the term…
Abstract
Compounds useful for treating inflammation, pain and swelling, represented by the formula: ##STR1## and the pharmaceutically acceptable acid addition salts thereof, wherein: Y and Z are each independently halo, alkyl or alkoxy; l and m are each independently integers of 0-4; b is an integer of 2-12; and X is selected from the group consisting of: --NR.sup.1 R.sup.2, --NR.sup.1 (CH.sub.2 CH.sub.2 OH), ##STR2## in which R.sup.1 and R.sup.2 are independently H, alkyl or cycloalkyl; R.sup.3 is H, alkyl or CH.sub.2 CH.sub.2 OH; and n is an integer of 3-7.
Claims15
A compound of the formula:
- ##STR17## and the pharmaceutically acceptable acid addition salts thereof, wherein:
- Y and Z are each independently halo, alkyl or alkoxy;
- l and m are each independently integers of 0-4;
- b is an integer of 2-12;
- and
- x is selected from the group consisting of:
- --NR.sup.1 R.sup.2, --NR.sup.1 (CH.sub.2 CH.sub.2 OH), ##STR18## in which R.sup.1 and R.sup.2 are each independently H, alkyl or cycloalkyl;
- R.sup.3 is H, alkyl or CH.sub.2 CH.sub.2 OH;
- and
- n is an integer of 3-7.
Dependencies are inferred from the claim text.