4-Amino-5-bromo-2-methoxy-N-[8-(benzyl)]-8-azabicyclo[3.2.1] -3-YL-benzamide or a pharmacologically acceptable acid addition salt thereof
AssigneeDelalande S.A.
InventorsPhilippe L. Dostert, Thierry F. Imbert, Bernard P. Bucher
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Abstract
There are disclosed nor-tropane derivatives substituted at the 3 position with aroylamino or heteroaroylamino and substituted at the 8 position with benzyl, substituted benzyl, 2-methyl thiophene, 3-methyl thiophene, 2-methyl furan or cyclohexylmethyl. The compounds are prepared by condensing the carboxylic acids corresponding to said aroyl or heteroaroyl group with the corresponding .beta.-3-amino-8-substituted nor-tropanes. The compounds possess neuroleptic properties.
Claims1
A compound having the formula ##STR85## wherein (I) ACO is 2-methoxy-4-amino-5-bromo benzoyl and R is ##STR86## or a pharmacologically acceptable acid addition salt thereof.
Dependencies are inferred from the claim text.