Antimycotic substituted 2,4-dichlorophenyl-imidazolyl-vinyl-carbinols
AssigneeBayer Aktiengesellschaft
InventorsWolf Reiser, Ludwig Elbe, Karl H. Buchel, Manfred Plempel
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Abstract
The invention relates to substituted 2,4-dichlorophenyl-imidazolyl-vinyl-carbinols of formula (I) as defined herein. The invention also includes methods for the manufacture of said compounds of formula (I), compositions containing said compounds of formula (I) and methods for the use of said compounds and compositions as antimycotic agents.
Claims16
A compound which is a substituted 2,4-dichlorophenyl-imidazolyl-vinyl carbinol of the formula ##STR17## or a salt thereof, in which
- R represents a cycloalkyl or cycloalkenyl radical which has in each case 5 to 7 carbon atoms and is optionally substituted by alkyl with 1 to 4 carbon atoms;
- a cycloalkyl-alkyl or cycloalkenylalkyl radical which has in each case 5 or 7 carbon atoms in the cycloalkyl or cycloalkenyl part and in each case 1 to 6 carbon atoms in the straight-chain or branched alkyl part and is optionally substituted by alkyl with 1 to 4 carbon atoms;
- an optionally substituted straight-chain or branched alkenyl or alkinyl radical with in each case up to 6 carbon atoms, the substituents being selected from:
- hydroxyl, alkoxy with 1 to 4 carbon atoms, and phenyl, which is optionally substituted by halogen or alkyl with 1 to 4 carbon atoms;
- phenyl substituted by phenoxy or chlorophenoxy;
- or optionally substituted phenylalkyl radical with 1 to 4 carbon atoms in the alkyl part in the racemic form and/or in the form of the geometric and/or optical isomers.
A compound which is 1-(2,4-dichlorophenyl)-2-(imidazol-1-yl)-4-ethyl-2-hexen-1-ol.
The compound which is 1-(2,4-dichlorophenyl)-2-(imidazol-1-yl)-2-penten-1-ol.
Dependencies are inferred from the claim text.