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US 4,241,071 AGranted
Antidepressant (.alpha.-phenyl-2-tolyl)azacycloalkanes
AssigneeAmerican Hoechst Corporation
InventorsLawrence L. Martin, Helen H. Ong, Vernon B. Anderson, Charles A. Crichlow
Life of this patent
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Abstract
Novel azacycloalkanes, azacycloalkenes and derivatives thereof and methods of preparing same are described. These compounds are useful as antidepressants, anticonvulsants, tranquilizers and analgetics.
Claims24
A compound of the formula ##STR19## wherein X is CH;
- Y is --(CH.sub.2).sub.n --;
- R is hydrogen, loweralkyl, phenylloweralkyl of the formula ##STR20## or cycloalkylloweralkyl in which the cycloalkyl portion contains from 3 to 6 carbon atoms;
- R.sup.1, R.sup.2 and R.sup.3 are the same or different and each can be hydrogen, halogen, alkoxy of from 1 to 2 carbon atoms, loweralkyl, hydroxy or trifluoromethyl;
- m is the integer 1 or 2;
- n is the integer 1, 2 or 3;
- the sum of m and n is 3 or 4;
- p is the integer 1, 2, 3 or 4;
- or a pharmaceutically acceptable acid addition salt thereof.
5 more elements
Dependencies are inferred from the claim text.