Substituted fluoracylresorcinols
AssigneeBoehringer Ingelheim GmbH
InventorsRolf Brickl, Hans Eberhardt, Karl-Richard Appel, Uwe Lechner, Walter Merk
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AssigneeBoehringer Ingelheim GmbH
InventorsRolf Brickl, Hans Eberhardt, Karl-Richard Appel, Uwe Lechner, Walter Merk
Estimating the term…
Compounds of the formula ##STR1## wherein R.sub.1 is perfluoroalkyl of 1 to 8 carbon atoms or 2,2,3,3-tetrafluoro-cyclobutyl, R.sub.2 and R.sub.4, which may be identical to or different from each other, are each hydrogen, alkyl of 1 to 10 carbon atoms, aliphatic acyl of 2 to 18 carbon atoms, benzoyl, salicyloyl or phenylacetyl, and R.sub.3 and R.sub.5, which may be identical to or different from each other, are each alkyl of 3 to 18 carbon atoms, halogen, nitro, p-toluenesulfonyl, cyclopentyl, cyclohexyl, cycloheptyl, cyclododecyl, methylcyclohexyl, dimethylcyclohexyl, benzyl, methylthio or ##STR2## where R.sub.1, R.sub.2 and R.sub.4 have the meanings previously defined, Q is --CH.sub.2 -- or --S--, and G is R.sub.5, as above defined, or Q is R.sub.3, as above defined, and G is --CH.sub.2 -- or --S--, R.sub.3 may, in addition, also be hydroxyl, methoxy, methyl or cyano, and R.sub.5 may also be methyl, or one of substituents R.sub.3 and R.sub.5 is hydrogen or ethyl when the other has the meanings defined above except hydrogen, or when R.sub.1 has the meanings defined above except trifluoromethyl, or when R.sub.2 and R.sub.4 have the meanings defined above except hydrogen or methyl. The compounds are useful as active ingredients in pharmaceutical, cosmetic and pesticidal compositions.
A compound of the formula ##STR33## wherein R.sub.1 is perfluoralkyl of 1 to 8 carbon atoms,
The method of inhibiting the growth of bacteria and fungi which comprises contacting said bacteria and fungi with a composition of claim 19.
Dependencies are inferred from the claim text.