Benzo [B]thienopyridines, process for their preparation and therapeutic compositions containing same
AssigneeParcor
InventorsDaniel Frehel, Jean-Pierre Maffrand
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AssigneeParcor
InventorsDaniel Frehel, Jean-Pierre Maffrand
Estimating the term…
This invention relates to compounds having the formula: ##STR1## in which: R.sup.1 represents hydrogen or a lower alkyl group; an aralkyl group optionally substituted on the aromatic nucleus with at least a halogen atom or a hydroxy, nitro, amino, cyano, carboxy, carboxamido, alkoxycarbonyl, lower alkyl, lower alkoxy or trifluoromethyl group; a nicotinyl group; an isonicotinyl group; a picolyl group; a furfuryl group; a 5-methyl-furfuryl group; a 2- or 3-thenyl group; a 5-methyl-2- or 3-thenyl group; or a 5-chloro-2-thenyl group; R.sup.2 represents hydrogen or a lower alkyl radical; and R.sup.3 and R.sup.4 represent each hydrogen, a halogen atom or a hydroxy, lower alkyl or lower alkoxy group, And their addition salts with inorganic or organic acids. Said new compounds have typically a therapeutically useful sedative and blood-platelet aggregation inhibiting activity.
A compound selected from the compounds having the formula:
Therapeutic composition having a sedative activity comprising an effective amount of an active compound selected from the compounds having the formula:
Therapeutic composition having a blood-platelet aggregation inhibiting activity comprising an effective amount of an active compound selected from the compounds having the formula:
Dependencies are inferred from the claim text.