Derivatives of 1,2-diphenyl-3,5-dioxo-4-n-butyl-pyrazolidine and process for making same
AssigneeAntonio Gallardo, S.A.
InventorsDavid J. Roberts, Jacinto M. Mauri
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Abstract
The present invention concerns novel therapeutic compounds having the formula: ##STR1## wherein R is a basic compound comprising 2-amino-4-methylpyridine or 2-amino-2-thiazoline, and methods of making this compound.
Claims24
A pharmaceutical composition having anti-inflammatory activity in humans as well as in other animals, said composition comprising a therapeutic compound having the formula:
- ##STR4## in which R is 2-amino-2-thiazoline having the formula:
- ##STR5## together with a non-toxic pharmaceutically acceptable carrier or diluent therefor, said therapeutic compound present in sufficient amount to exhibit said activity.
A pharmaceutical composition having analgesic activity in humans as well as in other animals, said composition comprising a therapeutic compound having the formula:
- ##STR6## in which R is 2-amino-2-thiazoline having the formula:
- ##STR7## together with a non-toxic pharmaceutically acceptable carrier or diluent therefor, said therapeutic compound present in sufficient amount to exhibit said activity.
A pharmaceutical composition having anti-pyretic activity in humans as well as in other animals, said composition comprising a therapeutic compound having the formula:
- ##STR8## in which R is 2-amino-2-thiazoline having the formula:
- ##STR9## together with a non-toxic pharmaceutically acceptable carrier or diluent therefor, said therapeutic compound present in sufficient amount to exhibit said activity.
A pharmaceutical composition for treating rheumatic diseases in humans as well as in other animals, said composition comprising a therapeutic compound having the formula:
- ##STR10## in which R is 2-amino-2-thiazoline having the formula:
- ##STR11## together with a non-toxic pharmaceutically acceptable carrier or diluent therefor, said therapeutic compound present in an effective amount for carrying out said treatment.
Dependencies are inferred from the claim text.