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US 4,065,465 AGranted
Process for the preparation of substituted trichloroacetamidine derivatives
AssigneeMerck & Co., Inc.
InventorGeorge H. Denny
Life of this patent
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Abstract
Substituted trichloroacetamidine derivatives are prepared by reacting an appropriately substituted amine with trichloroacetamidine or a trichloroacetimidate. The substituted amines are 3-aminomethyl indole and 2-acetoxy-3-phenoxy propylamine.
Claims3
A process for the preparation of a compound having the formula:
- ##STR2## wherein R is 3-indolylmethyl;
- which comprises treating a compound having the formula:
- ##STR3## wherein X is amino or loweralkoxy;
- with a compound having the formula:
- R--NH.sub.2
- wherein
- R is as previously defined, at from room temperature to 100.degree. C for from 30 minutes to 40 hours.
4 more elements
Dependencies are inferred from the claim text.